Pyridine-based, microwave-assisted one-pot synthetic protocol for the synthesis of ethyl 3-substituted-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carboxylates

被引：0
作者：
Sourabh Mundra
Radhakrishnan Mahesh
机构：
[1] Birla Institute of Technology and Science,Department of Pharmacy, FD
[2] Pilani,III
来源：
Research on Chemical Intermediates | 2016年 / 42卷
关键词：
5-Carboethoxy-2-thiouracil; Thiourea; Pyrimidine; Microwave irradiation; Synthesis;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Pyridine has been used for one-pot, two-component synthesis of ethyl 3-substituted-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carboxylate derivatives in moderate to good yields by condensing N-substituted thioureas with diethyl ethoxymalonate under microwave irradiation.
引用
收藏
页码：4207 / 4219
页数：12
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