Synthesis of new pyrido[4,3-e][1,2,4]triazolo-[5,1-c][1,2,4]triazin-6(7H)-ones

被引：0

作者：

Mohammad N. Mawlood

Mikhail A. Potapov

Irina V. Ledenyova

Oleg A. Kozaderov

Nadezhda V. Stolpovskaya

Khidmet S. Shikhaliev

Andrey Yu. Potapov

机构：

[1] Voronezh State University,

来源：

Chemistry of Heterocyclic Compounds | 2020年 / 56卷

关键词：

enamine; ethyl acetoacetate; dimethylformamide dimethyl acetal; hydrazone; pyrido[4,3-; ][1,2,4]triazolo[5,1-; ][1,2,4]triazine; 1,2,4-triazole-5-diazonium salt; [1,2,4]triazolo[5,1-; ][1,2,4]triazine;

D O I：

暂无

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学科分类号：

摘要：

Coupling of 3-substituted 1,2,4-triazole-5-diazonium salts with ethyl acetoacetate afforded 1,2,4-triazol-5-ylhydrazones, the reaction of which with dimethylformamide dimethyl acetal leads to the formation of the corresponding readily separable 4-[2-(dimethylamino)-vinyl][1,2,4]triazolo[5,1-c][1,2,4]triazine-3-carboxylates. New pyrido[4,3-e][1,2,4]triazolo[5,1-c][1,2,4]triazin-6(7H)-ones were synthesized by the condensation of the latter with primary amines.

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页码：1348 / 1352

页数：4

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