N-amination of unsymmetrically substituted pyrimidines. Synthesis of isomeric N-aminopyrimidones

被引：0

作者：

Bodyagin, M.B. ^{[1
]}

Ivanov, A.Yu. ^{[1
]}

Wurst, K. ^{[1
]}

Schantl, J.G. ^{[1
]}

Lobanov, P.S. ^{[1
]}

Potekhin, A.A. ^{[1
]}

机构：

[1] St. Petersburg State University, St. Petersburg 198904, Petrodvorets

来源：

Chemistry of Heterocyclic Compounds | 2003年 / 39卷 / 02期

关键词：

4-pyrimidones; N-amination; O-(mesitylenesulfonyl)hydroxylamine;

D O I：

10.1023/A:1023716424186

中图分类号：

学科分类号：

摘要：

N-Amination of 6-amino-2-methyl-4-pyrimidone with O-(mesitylenesulfonyl)hydroxylamine leads to the 3-amino derivative. The isomeric 1,6-diamino-2-methyl-4-pyrimidone was obtained by the N-amination of the O-benzoyl derivative of the initial pyrimidone and removal of the benzoyl protection.

引用

页码：195 / 199

页数：4