The First Example of 4,7,8,9-Tetrahydrothieno-[2,3-d]Azocine Synthesis by Domino Reaction of 4-ARYL-4,5,6,7-Tetrahydrothieno[3,2-c]Pyridines with Activated Alkynes

被引：0
作者：
L. G. Voskressensky
T. N. Borisova
T. M. Chervyakova
M. D. Matveeva
D. V. Galaktionova
S. V. Tolkunov
V. S. Tolkunova
A. B. Eresko
A. V. Varlamov
机构：
[1] People’s Friendship University of Russia,L. M. Litvinenko Institute of Physical
[2] Academy of Sciences of Ukraine,Organic Chemistry and Coal Chemistry
来源：
Chemistry of Heterocyclic Compounds | 2014年 / 50卷
关键词：
activated alkynes; tetrahydrothieno[2,3-; ]azocines; tetrahydrothieno[3,2-; ]pyridines; tetrahydropyridine ring expansion domino reaction;
D O I：
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中图分类号：
学科分类号：
摘要：
1-Aryl-substituted tetrahydrothieno[3,2-с]pyridines easily undergo domino reactions with activated alkynes, giving good yields of the corresponding tetrahydrothieno[2,3-d]azocines. The reactions of 1-methyl-substituted tetrahydrothieno[3,2-с]pyridine were more complicated.
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页码：1338 / 1345
页数：7
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