Endothelin-1 Binding to Endothelin Receptors in the Rat Anterior Pituitary Gland: Interaction in the Recognition of Endothelin-1 Between ETA and ETB Receptors

被引:13
|
作者
Akihiko Himeno [1 ]
Kazuto Shigematsu [2 ]
Takashi Taguchi [2 ]
Masami Niwa [1 ]
机构
[1] Nagasaki University School of Medicine,Department of Pharmacology 1
[2] Nagasaki University School of Medicine,Department of Pathology 2
关键词
endothelin ET; receptor; ET; receptor; cross-talk; endothelin-1; bivalent ligand; I-endothelin-l binding; quantitative receptor autoradiography; anterior pituitary gland (rat);
D O I
10.1023/A:1022557717481
中图分类号
学科分类号
摘要
1. 125I-Endothelin (ET)-1 binding to the rat anterior pituitary gland was saturable and single, with a Kd of 71 pM and a Bmax of 120 fmol/mg.
引用
收藏
页码:447 / 452
页数:5
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