Endothelin-1 Binding to Endothelin Receptors in the Rat Anterior Pituitary Gland: Interaction in the Recognition of Endothelin-1 Between ETA and ETB Receptors

被引：13
|
作者：
Akihiko Himeno [1 ]
Kazuto Shigematsu [2 ]
Takashi Taguchi [2 ]
Masami Niwa [1 ]
机构：
[1] Nagasaki University School of Medicine,Department of Pharmacology 1
[2] Nagasaki University School of Medicine,Department of Pathology 2
来源：
Cellular and Molecular Neurobiology | 1998年 / 18卷 / 4期
关键词：
endothelin ET; receptor; ET; receptor; cross-talk; endothelin-1; bivalent ligand; I-endothelin-l binding; quantitative receptor autoradiography; anterior pituitary gland (rat);
D O I：
10.1023/A:1022557717481
中图分类号：
学科分类号：
摘要：
1. 125I-Endothelin (ET)-1 binding to the rat anterior pituitary gland was saturable and single, with a Kd of 71 pM and a Bmax of 120 fmol/mg.
引用
收藏
页码：447 / 452
页数：5
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