Yap governs a lineage-specific neuregulin1 pathway-driven adaptive resistance to RAF kinase inhibitors

被引:0
作者
Maria E. R. Garcia-Rendueles
Gnana Krishnamoorthy
Mahesh Saqcena
Adrian Acuña-Ruiz
Giovanna Revilla
Elisa de Stanchina
Jeffrey A. Knauf
Rona Lester
Bin Xu
Ronald A. Ghossein
James A. Fagin
机构
[1] Memorial Sloan Kettering Cancer Center,Human Oncology and Pathogenesis Program
[2] IMDEA Food Institute,Antitumor Assessment Core Facility
[3] Memorial Sloan Kettering Cancer Center,Department of Medicine
[4] Memorial Sloan Kettering Cancer Center,Department of Pathology
[5] Memorial Sloan Kettering Cancer Center,undefined
[6] Weill-Cornell Medical College,undefined
来源
Molecular Cancer | / 21卷
关键词
Hippo; YAP; BRAF; Thyroid cancer; HER2; HER3; NRG1; Resistance; Dependency; Vemurafenib; Lapatinib;
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[1]  
Corcoran RB(2012)EGFR-mediated re-activation of MAPK signaling contributes to insensitivity of BRAF mutant colorectal cancers to RAF inhibition with vemurafenib Cancer Discov 2 227-235
[2]  
Montero-Conde C(2013)Relief of feedback inhibition of HER3 transcription by RAF and MEK inhibitors attenuates their antitumor effects in BRAF-mutant thyroid carcinomas Cancer Discov 3 520-533
[3]  
Prahallad A(2012)Unresponsiveness of colon cancer to BRAF(V600E) inhibition through feedback activation of EGFR Nature 483 100-103
[4]  
Poulikakos PI(2010)RAF inhibitors transactivate RAF dimers and ERK signalling in cells with wild-type BRAF Nature 464 427-430
[5]  
Yao Z(2015)BRAF mutants evade ERK-dependent feedback by different mechanisms that determine their sensitivity to pharmacologic inhibition Cancer Cell 28 370-383
[6]  
Lito P(2012)Relief of profound feedback inhibition of mitogenic signaling by RAF inhibitors attenuates their activity in BRAFV600E melanomas Cancer Cell 22 668-682
[7]  
Shalem O(2014)Genome-scale CRISPR-Cas9 knockout screening in human cells Science 343 84-87
[8]  
Lin L(2015)The Hippo effector YAP promotes resistance to RAF- and MEK-targeted cancer therapies Nat Genet 47 250-256
[9]  
Kapoor A(2014)Yap1 activation enables bypass of oncogenic Kras addiction in pancreatic cancer Cell 158 185-197
[10]  
Shao DD(2014)KRAS and YAP1 converge to regulate EMT and tumor survival Cell 158 171-184