Studies on antimicrobial activity for multidrug resistance strain by using phenyl pyrazolones substituted 3-(4-aminophenyl)-2-phenylquinazolin-4(3H)-one derivatives in vitro condition and their dyeing performance

被引：0
|
作者：
Nikhil Parekh
Kalpana Maheria
机构：
[1] S. V. National Institute of Technology,Applied Chemistry Department
来源：
Fibers and Polymers | 2012年 / 13卷
关键词：
3-(4-Aminophenyl)-2-phenylquinazolin-4(3H)-one; Phenyl pyrazolones; Synthesis; Antimicrobial activity; Dyeing; Fastness properties;
D O I：
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中图分类号：
学科分类号：
摘要：
Heterocyclic monoazo quinazolinone based azo dyes derived by the diazotization of 3-(4-aminophenyl)-2-phenylquinazolin-4(3H)-one with various phenyl pyrazolones based coupling components. All the heterocyclic azo dyes have been characterized by their percentage yield, UV-VIS spectroscopy, elemental analysis, IR spectroscopy, 1H NMR spectroscopy, and dyeing performance on silk, wool, nylon, and polyester fibers. All the dyes gave moderate to excellent fastness properties on each fiber. The main focus was to synthesize heterocyclic monoazo dyes that give good dyeing property along with pharmacological activity (anti bacterial and antifungal). Therefore, the synthesized compounds were examined for their antimicrobial activity at various concentrations using well-known Kirby-Bauer disk diffusion method.
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页码：162 / 168
页数：6
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