Synthesis and antimicrobial activity of some acridone derivatives bearing 1,3,4-oxadiazole moiety

被引：0
|
作者：
T. N. Kudryavtseva
P. I. Sysoev
S. V. Popkov
G. V. Nazarov
L. G. Klimova
机构：
[1] Kursk State University,
[2] D. I. Mendeleev Russian University of Chemistry and Technology,undefined
[3] Kursk State Medical University,undefined
来源：
Russian Chemical Bulletin | 2015年 / 64卷
关键词：
acridone; acridone acetic acid; hydrazide; 1,3,4-oxadiazole; antibacterial activity;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Novel acridone derivatives bearing 1,3,4-moiety were synthesized by intramolecular cyclization of N´-[2-(9-oxoacridin-10(9H)-yl)acetyl]arylhydrazides. Study of antimicrobial activity of the synthesized compounds reveals that some of them are more active than the comparator drug rivanol.
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页码：1341 / 1344
页数：3
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