Evaluation of some thiophene-based sulfonamides as potent inhibitors of carbonic anhydrase I and II isoenzymes isolated from human erythrocytes by kinetic and molecular modelling studies

被引：0
|
作者：
Zuhal Alım
Zeynep Köksal
Muhammet Karaman
机构：
[1] Kırşehir Ahi Evran University,Department of Chemistry, Faculty of Science and Arts
[2] Istanbul Medeniyet University,Department of Chemistry, Faculty of Engineering and Natural Sciences
[3] Kilis 7 Aralık University,Department of Molecular Biology and Genetics, Faculty of Arts and Sciences
来源：
Pharmacological Reports | 2020年 / 72卷
关键词：
Thiophene; Sulfonamide; Carbonic anhydrase; Inhibition; Molecular modelling;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：1738 / 1748
页数：10
相关论文
共 13 条
  • [11] Carbonic anhydrase inhibitors. Identification of selective inhibitors of the human mitochondrial isozymes VA and VB over the cytosolic isozymes I and II from a natural product-based phenolic library
    Davis, Rohan A.
    Innocenti, Alessio
    Poulsen, Sally-Ann
    Supuran, Claudiu T.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 18 (01) : 14 - 18
  • [12] Novel 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide based thiosemicarbazides as potent and selective inhibitors of tumor-associated human carbonic anhydrase IX and XII: Synthesis, cytotoxicity, and molecular modelling studies
    Demir-Yazici, Kubra
    Trawally, Muhammed
    Bua, Silvia
    Ozturk-Civelek, Dilek
    Akdemir, Atilla
    Supuran, Claudiu T.
    Guzel-Akdemir, Ozlen
    BIOORGANIC CHEMISTRY, 2024, 144
  • [13] Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors
    Mishra, Chandra Bhushan
    Kumari, Shikha
    Angeli, Andrea
    Monti, Simona Maria
    Buonanno, Martina
    Prakash, Amresh
    Tiwari, Manisha
    Supuran, Claudiu T.
    JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2016, 31 : 174 - 179
12