Evaluation of some thiophene-based sulfonamides as potent inhibitors of carbonic anhydrase I and II isoenzymes isolated from human erythrocytes by kinetic and molecular modelling studies

被引：0

作者：

Zuhal Alım

Zeynep Köksal

Muhammet Karaman

机构：

[1] Kırşehir Ahi Evran University,Department of Chemistry, Faculty of Science and Arts

[2] Istanbul Medeniyet University,Department of Chemistry, Faculty of Engineering and Natural Sciences

[3] Kilis 7 Aralık University,Department of Molecular Biology and Genetics, Faculty of Arts and Sciences

来源：

Pharmacological Reports | 2020年 / 72卷

关键词：

Thiophene; Sulfonamide; Carbonic anhydrase; Inhibition; Molecular modelling;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

引用

页码：1738 / 1748

页数：10

共 13 条

[1] Evaluation of some thiophene-based sulfonamides as potent inhibitors of carbonic anhydrase I and II isoenzymes isolated from human erythrocytes by kinetic and molecular modelling studies
Alim, Zuhal
Koksal, Zeynep
Karaman, Muhammet
PHARMACOLOGICAL REPORTS, 2020, 72 (06) : 1738 - 1748
[2] Inhibition properties of some flavonoids on carbonic anhydrase I and II isoenzymes purified from human erythrocytes
Huyut, Zubeyir
Beydemir, Sukru
Gulcin, Ilhami
JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY, 2017, 31 (09)
[3] Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors
Chiaramonte, Niccolo
Bua, Silvia
Angeli, Andrea
Ferraroni, Marta
Picchioni, Ilaria
Bartolucci, Gianluca
Braconi, Laura
Dei, Silvia
Teodori, Elisabetta
Supuran, Claudiu T.
Romanelli, Maria Novella
BIOORGANIC CHEMISTRY, 2019, 91
[4] Kinetic and in silico studies of hydroxy-based inhibitors of carbonic anhydrase isoforms I and II
Salmas, Ramin Ekhteiari
Mestanoglu, Mert
Durdagi, Serdar
Senturk, Murat
Kaya, A. Afsin
Kaya, Elif Celenk
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2016, 31 (01) : 31 - 37
[5] Inhibition Profiles of Some Symmetric Sulfamides Derived from Phenethylamines on Human Carbonic Anhydrase I, and II Isoenzymes
Topal, Fevzi
Aksu, Kadir
Gulcin, Ilhami
Tumer, Ferhan
Goksu, Suleyman
CHEMISTRY & BIODIVERSITY, 2021, 18 (10)
[6] Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and molecular docking studies
Eldehna, Wagdy M.
Al-Ansary, Ghada H.
Bua, Silvia
Nocentini, Alessio
Gratteri, Paola
Altoukhy, Ayman
Ghabbour, Hazem
Ahmed, Hanaa Y.
Supuran, Claudiu T.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 127 : 521 - 530
[7] Nimesulide linked acyl thioureas potent carbonic anhydrase I, II and α-glucosidase inhibitors: Design, synthesis and molecular docking studies
Ahmed, Atteeque
Sha, Imran
Saeed, Aamer
Shabir, Ghulam
Saleem, Arslan
Taslimi, Parham
Tok, Tugba Taskin
Kirici, Mahinur
Uc, Eda Mehtap
Hashmi, Muhammad Zaffar
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS, 2022, 6
[8] Kinetic and docking studies of phenol-based inhibitors of carbonic anhydrase isoforms I, II, IX and XII evidence a new binding mode within the enzyme active site
Durdagi, Serdar
Senturk, Murat
Ekinci, Deniz
Balaydin, Halis Turker
Goksu, Suleyman
Kufrevioglu, O. Irfan
Innocenti, Alessio
Scozzafava, Andrea
Supuran, Claudiu T.
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 19 (04) : 1381 - 1389
[9] Identification of the Inhibition Effects of Some Natural Antiproliferative Agents on CA-I, CA-II, and AChE Activities Isolated from Human Erythrocytes by Kinetic and Molecular Docking Studies
Kilinc, N.
Guller, U.
Alim, Z.
RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY, 2022, 48 (04) : 720 - 730
[10] Identification of the Inhibition Effects of Some Natural Antiproliferative Agents on CA-I, CA-II, and AChE Activities Isolated from Human Erythrocytes by Kinetic and Molecular Docking Studies
N. Kılınç
U. Güller
Z. Alım
Russian Journal of Bioorganic Chemistry, 2022, 48 : 720 - 730

← 1 2 →