Hit-to-lead optimization of amino-carboxamide benzothiazoles as LSD1 inhibitors

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作者
Du’a Al bustanji
Soraya Alnabulsi
Enas A. Al-Hurani
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[1] Jordan University of Science and Technology,Department of Medicinal Chemistry and Pharmacognosy, Faculty of Pharmacy
[2] P.O. Box 3030,undefined
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LSD1 enzyme; hit-to-lead optimization; anticancer; structure-activity relationship; amino-carboxamide benzothiazoles.;
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页码:910 / 929
页数:19
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