Prenylation inhibitors stimulate both estrogen receptor α transcriptional activity through AF-1 and AF-2 and estrogen receptor β transcriptional activity

被引:0
作者
Philippe Cestac
Guillaume Sarrabayrouse
Claire Médale-Giamarchi
Philippe Rochaix
Patrick Balaguer
Gilles Favre
Jean-Charles Faye
Sophie Doisneau-Sixou
机构
[1] INSERM U563 and Institut Claudius Regaud,Département 'Innovation Thérapeutique et Oncologie Moléculaire', Centre de Physiopathologie de Toulouse Purpan
[2] Endocrinologie Moléculaire et Cellulaire des Cancers,INSERM 540
来源
Breast Cancer Research | / 7卷
关键词
estrogen receptor; farnesyltransferase inhibitor; geranylgeranyltransferase inhibitor; Rho proteins; transcription;
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