In vitro and in vivo characterization of JNJ-31020028 (N-(4-{4-[2-(diethylamino)-2-oxo-1-phenylethyl]piperazin-1-yl}-3-fluorophenyl)-2-pyridin-3-ylbenzamide), a selective brain penetrant small molecule antagonist of the neuropeptide Y Y2 receptor

被引：0
|
作者：
James R. Shoblock
Natalie Welty
Diane Nepomuceno
Brian Lord
Leah Aluisio
Ian Fraser
S. Timothy Motley
Steve W. Sutton
Kirsten Morton
Ruggero Galici
John R. Atack
Lisa Dvorak
Devin M. Swanson
Nicholas I. Carruthers
Curt Dvorak
Timothy W. Lovenberg
Pascal Bonaventure
机构：
[1] Johnson & Johnson Pharmaceutical Research and Development,
[2] L.L.C.,undefined
来源：
Psychopharmacology | 2010年 / 208卷
关键词：
Neuropeptide Y Y; receptor; Norepinephrine; Microdialysis; Stress-induced anorexia; Hypothalamus; Anxiety;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：265 / 277
页数：12
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