Direct Comparison of [18F]F-DPA with [18F]DPA-714 and [11C]PBR28 for Neuroinflammation Imaging in the same Alzheimer’s Disease Model Mice and Healthy Controls

[1] Guilarte TR(1995)Enhanced expression of peripheral benzodiazepine receptors in trimethyltin-exposed rat brain: a biomarker of neurotoxicity Neurotoxicology 16 441-450

[2] Kuhlmann AC(1989)Synthesis and evaluation of Ann Nucl Med 3 63-71

[3] O'Callaghan JP(2008)C-PK 11195 for in vivo study of peripheral-type benzodiazepine receptors using positron emission tomography J Nucl Med 49 814-822

[4] Miceli RC(2019)DPA-714, a new translocator protein-specific ligand: synthesis, radiofluorination, and pharmacologic characterization Alzheimer's Dement 15 1081-1103

[5] Hashimoto K(2004)A new perspective for advanced positron emission tomography-based molecular imaging in neurodegenerative proteinopathies Neurochem Int 44 433-440

[6] Inoue O(2003)Evaluation of three quinoline-carboxamide derivatives as potential radioligands for the in vivo PET imaging of neurodegeneration Nucl Med Biol 30 199-206

[7] Suzuki K(2009)The peripheral benzodiazepine receptor ligand PK11195 binds with high affinity to the acute phase reactant alpha1-acid glycoprotein: implications for the use of the ligand as a CNS inflammatory marker J Med Chem 52 688-699

[8] Yamasaki T(2012)Single-step high-yield radiosynthesis and evaluation of a sensitive Bioorg Med Chem Lett 22 1308-1313

[9] Kojima M(2020)F-labeled ligand for imaging brain peripheral benzodiazepine receptors with PET J Cereb Blood Flow Metab 40 1012-1020

[10] James ML(2018)[ Nucl Med Biol 67 1-6

[1] Guilarte TR(1995)Enhanced expression of peripheral benzodiazepine receptors in trimethyltin-exposed rat brain: a biomarker of neurotoxicity Neurotoxicology 16 441-450

[2] Kuhlmann AC(1989)Synthesis and evaluation of Ann Nucl Med 3 63-71

[3] O'Callaghan JP(2008)C-PK 11195 for in vivo study of peripheral-type benzodiazepine receptors using positron emission tomography J Nucl Med 49 814-822

[4] Miceli RC(2019)DPA-714, a new translocator protein-specific ligand: synthesis, radiofluorination, and pharmacologic characterization Alzheimer's Dement 15 1081-1103

[5] Hashimoto K(2004)A new perspective for advanced positron emission tomography-based molecular imaging in neurodegenerative proteinopathies Neurochem Int 44 433-440

[6] Inoue O(2003)Evaluation of three quinoline-carboxamide derivatives as potential radioligands for the in vivo PET imaging of neurodegeneration Nucl Med Biol 30 199-206

[7] Suzuki K(2009)The peripheral benzodiazepine receptor ligand PK11195 binds with high affinity to the acute phase reactant alpha1-acid glycoprotein: implications for the use of the ligand as a CNS inflammatory marker J Med Chem 52 688-699

[8] Yamasaki T(2012)Single-step high-yield radiosynthesis and evaluation of a sensitive Bioorg Med Chem Lett 22 1308-1313

[9] Kojima M(2020)F-labeled ligand for imaging brain peripheral benzodiazepine receptors with PET J Cereb Blood Flow Metab 40 1012-1020

[10] James ML(2018)[ Nucl Med Biol 67 1-6