4-Hydroxy-2-quinolones. 90.* Synthesis and antitubercular activity of 4-methyl-2-thiazolylamides of halo-substituted 4-hydroxy-2-oxo-1,2-dihydro-3- quinolinecarboxylic acids

被引：0

作者：

Ukrainets I.V. ^{[1
]}

Sidorenko L.V. ^{[1
]}

Petrushova L.A. ^{[1
]}

Gorokhova O.V. ^{[1
]}

机构：

[1] National Pharmaceutical University

来源：

Chemistry of Heterocyclic Compounds | 2006年 / 42卷 / 1期

关键词：

2-amino-4-methylthiazole; 4-hydroxy-2-oxo-1,2-dihydro-3- quinolinecarboxylic acids; Amides; Antitubercular activity;

D O I：

10.1007/s10593-006-0048-8

中图分类号：

学科分类号：

摘要：

Several variants were studied for the synthesis of esters of halogen derivatives of 4-hydroxy-2-oxo-1,2-dihydro-3-quinolinecarboxylic acids, whose reaction with 2-amino-4-methylthiazole gives the corresponding hetarylamides. Results are given for a study of the antitubercular activity of these products. ©2006 Springer Science+Business Media, Inc.

引用

页码：64 / 69

页数：5

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