Catalyst-free tandem Michael addition-cyclization reactions in aqueous media for the synthesis of benzimidazo[1,2-a]pyrimidinone derivatives

被引:0
作者
ChuanLi Ren
Yan Wang
Dong Wang
YongJun Chen
Li Liu
机构
[1] Chinese Academy of Sciences,Beijing National Laboratory (BNLMS), CAS Key Laboratory for Molecular Recognition and Function
[2] Chinese Academy of Sciences,Institute of Chemistry
来源
Science China Chemistry | 2010年 / 53卷
关键词
queous media; Baylis-Hillman alcohol; 2-aminobenzimidazole; pesticidal activity;
D O I
暂无
中图分类号
学科分类号
摘要
The catalyst-free reactions of Baylis-Hillman alcohols (1a-i) with 2-aminobenzimidazole (2) in THF-H2O (1:4) were developed for the convenient and greener synthesis of benzimidazo[1,2-a]pyrimidinone derivatives (3a-i). The pesticidal activities of 3a-i were examined to investigate a new biological activity of the imidazo[1,2-a]pyrimidinone-type compounds.
引用
收藏
页码:1492 / 1496
页数:4
相关论文
共 96 条
  • [91] Hu L.Q.(undefined)undefined undefined undefined undefined-undefined
  • [92] Ranu B.C.(undefined)undefined undefined undefined undefined-undefined
  • [93] Banerjee S.(undefined)undefined undefined undefined undefined-undefined
  • [94] Brindaban C.(undefined)undefined undefined undefined undefined-undefined
  • [95] Ranu S.(undefined)undefined undefined undefined undefined-undefined
  • [96] Banerjee undefined(undefined)undefined undefined undefined undefined-undefined