The endomorphin-1/2 and dynorphin-B peptides display biased agonism at the mu opioid receptor

被引:0
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作者
Justin LaVigne
Attila Keresztes
Daniel Chiem
John M. Streicher
机构
[1] University of Arizona,Department of Pharmacology, College of Medicine
[2] University of New England,Department of Biomedical Sciences, College of Osteopathic Medicine
来源
Pharmacological Reports | 2020年 / 72卷
关键词
Endogenous opioid peptides; Endomorphin; Biased agonism; Forskolin-stimulated cAMP accumulation; S-GTPγS coupling;
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页码:465 / 471
页数:6
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