Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells

被引:0
|
作者
Yue-qin Wang
Ai-jun Shen
Jing-ya Sun
Xin Wang
Hong-chun Liu
Min-min Zhang
Dan-qi Chen
Bing Xiong
Jing-kang Shen
Mei-yu Geng
Min Zheng
Jian Ding
机构
[1] China Pharmaceutical University,Department of New Drug Screening Center
[2] Division of Anti-tumor Pharmacology,Department of Thoracic Surgery
[3] Synthetic Organic and Medicinal Chemistry Laboratory,undefined
[4] State Key Laboratory of Drug Research,undefined
[5] Shanghai Institute of Materia Medica,undefined
[6] Chinese Academy of Sciences,undefined
[7] Shanghai Tongren Hospital,undefined
[8] Shanghai Jiao Tong University School of Medicine,undefined
来源
Acta Pharmacologica Sinica | 2016年 / 37卷
关键词
non-small cell lung cancer; gefitinib resistance; Hsp90;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:1587 / 1596
页数:9
相关论文
共 50 条
  • [1] Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells
    Wang, Yue-qin
    Shen, Ai-jun
    Sun, Jing-ya
    Wang, Xin
    Liu, Hong-chun
    Zhang, Min-min
    Chen, Dan-qi
    Xiong, Bing
    Shen, Jing-kang
    Geng, Mei-yu
    Zheng, Min
    Ding, Jian
    ACTA PHARMACOLOGICA SINICA, 2016, 37 (12) : 1587 - 1596
  • [3] Novel Hsp90 Inhibitor C086 Potently Inhibits Non-Small Cell Lung Cancer Cells As A Single Agent Or In Combination With Gefitinib
    Wang, Liman
    Fan, Yingjuan
    Mei, Hanhao
    Liu, Yang
    Zhang, Lianru
    Xu, Jianhua
    Huang, Xuhui
    CANCER MANAGEMENT AND RESEARCH, 2019, 11 : 8937 - 8945
  • [4] Management of EGFR-Mutant Non-Small Cell Lung Cancer: Focus on Gefitinib
    Naito, Yoichi
    Goto, Koichi
    CLINICAL MEDICINE INSIGHTS-THERAPEUTICS, 2009, 1 : 1027 - 1040
  • [5] The HSP90 inhibitor ganetespib potentiates the antitumor activity of EGFR tyrosine kinase inhibition in mutant and wild-type non-small cell lung cancer
    Smith, Donald L.
    Acquaviva, Jaime
    Sequeira, Manuel
    Jimenez, John-Paul
    Zhang, Chaohua
    Sang, Jim
    Bates, Richard C.
    Proia, David A.
    TARGETED ONCOLOGY, 2015, 10 (02) : 235 - 245
  • [6] Synergistic activity of the Hsp90 inhibitor ganetespib with taxanes in non-small cell lung cancer models
    Proia, David A.
    Sang, Jim
    He, Suqin
    Smith, Donald L.
    Sequeira, Manuel
    Zhang, Chaohua
    Liu, Yuan
    Ye, Shuxia
    Zhou, Dan
    Blackman, Ronald K.
    Foley, Kevin P.
    Koya, Keizo
    Wada, Yumiko
    INVESTIGATIONAL NEW DRUGS, 2012, 30 (06) : 2201 - 2209
  • [7] Discovery of hybrid Hsp90 inhibitors and their anti-neoplastic effects against gefitinib-resistant non-small cell lung cancer (NSCLC)
    Jeong, Chul-Ho
    Park, Hee Baek
    Jang, Won Jun
    Jung, Su Hyun
    Seo, Young Ho
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (01) : 224 - 227
  • [8] The HSP90 inhibitor ganetespib potentiates the antitumor activity of EGFR tyrosine kinase inhibition in mutant and wild-type non-small cell lung cancer
    Donald L. Smith
    Jaime Acquaviva
    Manuel Sequeira
    John-Paul Jimenez
    Chaohua Zhang
    Jim Sang
    Richard C. Bates
    David A. Proia
    Targeted Oncology, 2015, 10 : 235 - 245
  • [9] PHASE II ACTIVITY OF THE HSP90 INHIBITOR AUY922 IN PATIENTS WITH EGFR-MUTANT ADVANCED NON-SMALL CELL LUNG CANCER (NSCLC
    Barlesi, Fabrice
    Besse, Benjamin
    Chu, Quincy
    Gandhi, Leena
    Griesinger, Frank
    Felip, Enriqueta
    Kang, Jin Hyoung
    Kim, Sang-We
    Rosell, Rafael
    Sequist, Lecia V.
    Soo, Ross
    Wallmark, John
    Avsar, Emin
    Ofosu-Appiah, William
    Pain, Scott
    Akimov, Mikhail
    Garon, Edward B.
    JOURNAL OF THORACIC ONCOLOGY, 2013, 8 : S611 - S612
  • [10] Celastrol Induces Apoptosis in Gefitinib-Resistant Non-Small Cell Lung Cancer Cells via Caspases-Dependent Pathways and Hsp90 Client Protein Degradation
    Fan, Xing-Xing
    Li, Na
    Wu, Jian-Lin
    Zhou, Yan-Ling
    He, Jian-Xing
    Liu, Liang
    Leung, Elaine Lai-Han
    MOLECULES, 2014, 19 (03): : 3508 - 3522