Synthesis, molecular docking, and in silico ADME prediction of some fused pyrazolo[1,5-a]pyrimidine and pyrazole derivatives as potential antimicrobial agents

被引：0
|
作者：
Ashraf S. Hassan
Nesrin M. Morsy
Hassan M. Awad
Ahmed Ragab
机构：
[1] National Research Centre,Organometallic and Organometalloid Chemistry Department
[2] National Research Centre,Chemistry of Natural and Microbial Products Department, Pharmaceutical and Drug Industries Research Division
[3] Al-Azhar University,Department of Chemistry, Faculty of Science (Boys)
来源：
Journal of the Iranian Chemical Society | 2022年 / 19卷
关键词：
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：521 / 545
页数：24
相关论文
共 50 条
  • [41] Preparation of some novel 3,5-diaminopyrazole, pyrazolo-[1,5-a][1,3,5]triazine and pyrazolo[1,5-a]-pyrimidine derivatives containing sulfonamido moieties as antimicrobial agents
    El-Gaby, MSA
    Taha, NM
    Micky, JA
    El-Sharief, MAMS
    ACTA CHIMICA SLOVENICA, 2002, 49 (01) : 159 - 171
  • [42] SYNTHESIS OF FUSED PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES UNDER MICROWAVE IRRADIATION AND ULTRASOUND, AS ECOFRIENDLY ENERGY SOURCES
    Al-Zaydi, Khadijah M.
    HETEROCYCLES, 2009, 78 (08) : 2003 - 2012
  • [43] Design, Synthesis, and Evaluation of the Anticancer Properties of a Novel Series of Imidazolone Fused Pyrazolo[1,5-a]pyrimidine Derivatives
    Kumar, Ajeesh A. K.
    Bodke, Yadav D.
    Gowda, Ashwath N.
    Sambasivam, Ganesh
    Bhat, Kishore G.
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2017, 54 (03) : 1904 - 1924
  • [44] Synthesis and NMR-spectroscopic investigation of pyrazolo[1,5-a]pyrimidine derivatives
    Makarov, VA
    Solovyeva, NP
    Granik, VG
    KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII, 1997, (05): : 619 - 628
  • [45] New One-Step Synthesis of Pyrazolo[1,5-a]pyrimidine and Pyrazolo[1,5-a]quinazoline Derivatives via Multicomponent Reactions
    Ghotekar, Bhausaheb K.
    Jachak, Madhukar N.
    Toche, Raghunath B.
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2009, 46 (04) : 708 - 713
  • [46] Design, Synthesis, and Characterization of Some Novel Pyrazolo [1,5-a] Pyrimidines as Potent Antimicrobial Agents
    Dawane, Bhaskar S.
    Konda, Shankaraiah G.
    Zangade, Sainath B.
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2010, 47 (05) : 1250 - 1254
  • [47] STUDIES WITH POLYFUNCTIONALLY SUBSTITUTED HETEROCYCLES - NOVEL SYNTHESIS OF PYRAZOLO[1,5-A]PYRIMIDINE, TRIAZOLO-[1,5-A]PYRIMIDINE AND PYRANOOXAZOLE DERIVATIVES
    KANDEEL, ZE
    FARAG, AM
    NEGM, AM
    KHALAFALL, AK
    RASSLAN, MAM
    ELNAGDI, MH
    JOURNAL OF CHEMICAL RESEARCH-S, 1994, (11): : 416 - 417
  • [48] Routes to pyrazolo[3,4-e][1,4]thiazepine, pyrazolo[1,5-a]pyrimidine and pyrazole derivatives
    Abu Elmaati, TM
    El-Taweel, FMA
    JOURNAL OF THE CHINESE CHEMICAL SOCIETY, 2003, 50 (3A) : 413 - 418
  • [49] Pyrazole clubbed triazolo[1,5-a]pyrimidine hybrids as an anti-tubercular agents: Synthesis, in vitro screening and molecular docking study
    Bhatt, Jaimin D.
    Chudasama, Chaitanya J.
    Patel, Kanuprasad D.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (24) : 7711 - 7716
  • [50] Synthesis and solvatochromic properties of some disazo dyes derived from pyrazolo[1,5-a]pyrimidine derivatives
    Tsai, PC
    Wang, IJ
    DYES AND PIGMENTS, 2005, 64 (03) : 259 - 264
12345