Palladium-Catalyzed Amination and Amidation of Benzo-Fused Bromine-Containing Heterocycles

被引：0

作者：

A. G. Sergeev

G. A. Artamkina

V. S. Velezheva

I. N. Fedorova

I. P. Beletskaya

机构：

[1] Lomonosov Moscow State University,Faculty of Chemistry

[2] Russian Academy of Sciences,Nesmeyanov Institute of Organometallic Compounds

来源：

Russian Journal of Organic Chemistry | 2005年 / 41卷

关键词：

Organic Chemistry; Palladium; Biphenyl; Catalytic System; Carbazole;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

Amination and amidation of bromoindole, 6-bromo-1,2,3,4-tetrahydrocarbazol-1-one, and 8-bromo-2,4,5,6-tetrahydro-1H-pyrazino[3,2,1-jk]carbazole derivatives was effected in the presence of palladium complexes. The use of the catalytic system Pd2dba3⋅CHCl3-2-[di(tert-butyl)phosphino]biphenyl in the amination and of Pd2dba3⋅CHCl3-Xantphos [or 3,5-(CF3)2Xantphos] in the amidation ensured moderate to high yields of the corresponding products.

引用

页码：860 / 874

页数：14

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