Peptide Blocker of Ion Channel TRPV1 Exhibits a Long Analgesic Effect in the Heat Stimulation Model

被引：0
|
作者：
O. V. Sintsova
V. A. Palikov
Y. A. Palikova
A. A. Klimovich
I. N. Gladkikh
Y. A. Andreev
M. M. Monastyrnaya
E. P. Kozlovskaya
I. A. Dyachenko
S. A. Kozlov
E. V. Leychenko
机构：
[1] Elyakov Pacific Institute of Bioorganic Chemistry,
[2] Far Eastern Branch,undefined
[3] Russian Academy of Sciences,undefined
[4] Shemyakin–Ovchinnikov Institute of Bioorganic Chemistry,undefined
[5] Pushchino Branch,undefined
[6] Russian Academy of Sciences,undefined
[7] Shemyakin–Ovchinnikov Institute of Bioorganic Chemistry,undefined
[8] Russian Academy of Sciences,undefined
[9] Institute of Molecular Medicine,undefined
[10] Sechenov First Moscow State Medical University,undefined
来源：
Doklady Biochemistry and Biophysics | 2020年 / 493卷
关键词：
sea anemone; TRPV1; nociception; analgesia;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：215 / 217
页数：2
相关论文
共 50 条
  • [41] Inhibitory effect of positively charged triazine antagonists of prokineticin receptors on the transient receptor vanilloid type-1 (TRPV1) channel
    De Petrocellis, Luciano
    Moriello, Aniello Schiano
    Byun, Joon Seok
    Sohn, Joo Mi
    Lee, Jae Yeol
    Vazquez-Romero, Ana
    Garrido, Maria
    Messeguer, Angel
    Zhang, Fang-Xiong
    Zamponi, Gerald W.
    Deplano, Alessandro
    Congiu, Cenzo
    Onnis, Valentina
    Balboni, Gianfranco
    Di Marzo, Vincenzo
    PHARMACOLOGICAL RESEARCH, 2015, 99 : 362 - 369
  • [42] Vanilloid TRPV1 receptor mediates the antihyperalgesic effect of the nonpsychoactive cannabinoid, cannabidiol, in a rat model of acute inflammation
    Costa, B
    Giagnoni, G
    Franke, C
    Trovato, AE
    Colleoni, M
    BRITISH JOURNAL OF PHARMACOLOGY, 2004, 143 (02) : 247 - 250
  • [43] Inhibitions of anandamide transport and FAAH synthesis decrease apoptosis and oxidative stress through inhibition of TRPV1 channel in an in vitro seizure model
    Mustafa Nazıroğlu
    Afife Nur Taner
    Esra Balbay
    Bilal Çiğ
    Molecular and Cellular Biochemistry, 2019, 453 : 143 - 155
  • [44] The Pain Pathway in the Rat following Noxious Thermal Stimulation: Effect of Morphine on pERK1/2 and TRPV1 at the Dorsal Horn Level, and on Hyperalgesia
    Donnerer, Josef
    Liebmann, Ingrid
    PHARMACOLOGY, 2013, 92 (1-2) : 32 - 38
  • [45] Acid-Sensing Ion Channel 3, But Not Capsaicin Receptor TRPV1, Plays a Protective Role in Isoproterenol-Induced Myocardial Ischemia in Mice
    Cheng, Ching-Feng
    Chen, I-Lun
    Cheng, Mei-Hsin
    Lian, Wei-Shiung
    Lin, Chao-Chieh
    Kuo, Terry B. J.
    Chen, Chih-Cheng
    CIRCULATION JOURNAL, 2011, 75 (01) : 174 - 178
  • [46] MOK, a pharmacopuncture medicine, regulates thyroid dysfunction in L-thyroxin-induced hyperthyroidism in rats through the regulation of oxidation and the TRPV1 ion channel
    Hwang, Ji Hye
    Kang, Seok Yong
    Kang, An Na
    Jung, Hyo Won
    Jung, Chul
    Jeong, Jin-Ho
    Park, Yong-Ki
    BMC COMPLEMENTARY AND ALTERNATIVE MEDICINE, 2017, 17
  • [47] The effect of Ma-Xin-Gan-Shi decoction on asthma exacerbated by respiratory syncytial virus through regulating TRPV1 channel
    Li, Mengwen
    Fan, Xinsheng
    Zhou, Liping
    Jiang, Minyue
    Shang, Erxin
    JOURNAL OF ETHNOPHARMACOLOGY, 2022, 291
  • [48] Effect of San'ao decoction with scorpio and bombyx batryticatus on CVA mice model via airway inflammation and regulation of TRPA1/TRPV1/TRPV5 channels
    Wang, Pengli
    Shang, Erxin
    Fan, Xinsheng
    JOURNAL OF ETHNOPHARMACOLOGY, 2021, 264
  • [49] Effects of activation of skin ion channels TRPM8, TRPV1, and TRPA1 on the immune response. Comparison with effects of cold and heat exposure
    Kozyreva, T., V
    Khramova, G. M.
    JOURNAL OF THERMAL BIOLOGY, 2020, 93
  • [50] Co-administration of transient receptor potential vanilloid 4 (TRPV4) and TRPV1 antagonists potentiate the effect of each drug in a rat model of cystitis
    Charrua, Ana
    Cruz, Celia D.
    Jansen, Dick
    Rozenberg, Boy
    Heesakkers, John
    Cruz, Francisco
    BJU INTERNATIONAL, 2015, 115 (03) : 452 - 460
12345