Regioisomeric acetoxy derivatives of 8-aza-D-homogona-12,17a-dione. Annelation of 1-methyl-3,4-dihydroisoquinoline with 4-acetoxy-2- acetylcyclohexane-1,3-dione

被引：0

作者：

Gulyakevich O.V. ^{[1
]}

Zaitsev V.G. ^{[1
]}

Mikhal'chuk A.L. ^{[1
]}

机构：

[1] Institute of Bioorganic Chemistry, National Academy of Sciences

来源：

Chemistry of Heterocyclic Compounds | 2004年 / 40卷 / 3期

关键词：

2-acylcyclohexane-1,3-diones; 3,4-dihydroisoquinolines; 8-aza-D-homogonanes; 8-azasteroids; Annelation; Cyclic Schiffs bases; Regioselectivity; Stereochemistry;

D O I：

10.1023/B:COHC.0000028627.77366.49

中图分类号：

学科分类号：

摘要：

Annelation ([2+4] cyclocondensation) of 1-methyl-3,4-dihydroisoquinoline with 4-acetoxy-2-acetylcyclohexane-1,2-dione leads to a mixture of regioisomeric acetoxy derivatives of 9-methyl-8-aza-D-homogona-12,17a-dione.

引用

页码：315 / 319

页数：4

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