Synthesis of piperine–amino acid ester conjugates and study of their cytotoxic activities against human cancer cell lines

被引:0
作者
V. Rama Subba Rao
G. Suresh
R. Ranga Rao
K. Suresh Babu
G. Chashoo
A. K. Saxena
J. Madhusudana Rao
机构
[1] Indian Institute of Chemical Technology,Division of Organic Chemistry
[2] Indian Institute of Integrative Medicine (CSIR),I, Natural Product Laboratory
来源
Medicinal Chemistry Research | 2012年 / 21卷
关键词
Piperine; Piperoic acid; Amino acid conjugates; Amide linkage; Peptide linkage; Boric acid; Cytotoxic activity;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:38 / 46
页数:8
相关论文
共 162 条
[1]  
Bezerra DP(2006)In vivo growth-inhibition of Sarcoma 180 By piplartine and piperine, two alkaloid amides from J Med Biol Res 39 801-807
[2]  
Castro FO(1985)Increased life expectancy resulting from addition of L-deprenyl to Madopar treatment in Parkinson’s disease: a longterm study J Neural Transm 64 113-127
[3]  
Alves APNN(2005)Plants as a source of anti-cancer agents J Ethnopharmacol 100 72-79
[4]  
Pessoa C(2009)Impact of natural products on developing new anti-cancer agents Chem Rev 109 3012-3043
[5]  
Moraes MO(2003)Apoptosis-based drug screening and detection of Selective toxicity to cancer cells Anti Cancer Drugs 14 555-561
[6]  
Silveira ER(2009)Diferuloylmethane augments the cytotoxic effects of piplartine isolated from Toxicol In Vitro 23 1085-1091
[7]  
Lima MAS(2005)Synthesis and biological activity of fluoroquinolonepyrrolo[2, 1-c][1, 4]benzodiazepine conjugates Bioorg Med Chem 13 2021-2029
[8]  
Elmiro FJM(2005)The evolving role of natural products in drug discovery Nat Rev Drug Discov. 4 206-220
[9]  
Costa-Lotufo LV(2004)Inhibition of MAO A and B by some plant-derived alkaloids, phenols and anthraquinones J Ethnopharmacol 91 351-355
[10]  
Birkmayer W(2006)Oncology exploration: charting cancer medicinal chemistry space Drug Discov Today 11 149-159