Synthesis of (2R,4R)-2-alkyl-3-(2-mercaptobenzoyl)thiazolidine-4-carboxylic acids

被引：0
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作者：
А. Yu. Ershov
I. V. Lagoda
D. G. Nasledov
M. Yu. Vasil’eva
L. Yu. Kuleshova
L. V. Pavlova
A. V. Yakimanskii
机构：
[1] Russian Academy of Sciences,Institute of Macromolecular Compounds
[2] Russian Ministry of Defense,R&D Test Center (of Medico
[3] Ryazan Medical University,Biological Protection), State R&D Institute of Military Medicine
[4] St. Petersburg State University,undefined
来源：
Russian Journal of Organic Chemistry | 2017年 / 53卷
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摘要：
Basing on natural amino acid L-cysteine, commercially available aliphatic aldehydes, 2-acetylsulfanylbenzoyl chloride and 2,2′-disulfandiyldibenzoyl dichloride a synthesis was developed of (2R,4R)-2-alkyl-3-(2-mercaptobenzoyl)thiazolidine-4-carboxylic acids, potential antihypertensive compounds, inhibitors of angiotensin transforming enzyme.
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页码：1682 / 1686
页数：4
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