Facile and efficient synthesis of functionalized iminothiopyran and isothiochromen via one-pot multicomponent reactions

被引：0
作者：
Hosein Hamadi
Mehdi Khoobi
Zinatossadat Hossaini
Abbas Shafiee
机构：
[1] Tarbiat Modares University,Department of Chemistry
[2] Zanjan University,Department of Chemistry
[3] Islamic Azad University,Chemistry Department
[4] Tehran University of Medical Sciences,Department of Chemistry, Faculty of Pharmacy, and Pharmaceutical Sciences Research Center
来源：
Molecular Diversity | 2011年 / 15卷
关键词：
6; -6-iminothiopyran-2,3-dicarboxylate; Aryl isothiocyanate; Dialkyl acetylenedicarboxylate; 1; -isothiochromene-3,4-dicarboxylate; Multicomponent reaction; MCR;
D O I：
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中图分类号：
学科分类号：
摘要：
An efficient synthesis of 6H-6-iminothiopyran-2,3-dicarboxylate and 1H-isothiochromene-3,4-dicarboxylate derivatives via one-pot reactions between acetylenic esters, aryl isothiocyanates and enaminones in dichloromethane at room temperature is described. The mild reaction condition, high yields and the new products are advantages of our method.
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页码：35 / 40
页数：5
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