Effect of ceritinib on the pharmacokinetics of coadministered CYP3A and 2C9 substrates: a phase I, multicenter, drug–drug interaction study in patients with ALK + advanced tumors

被引:1
作者
Felipe K. Hurtado
Filippo de Braud
Javier De Castro Carpeño
Maria Jose de Miguel Luken
Ding Wang
Jeffrey Scott
Yvonne Y. Lau
Tracey McCulloch
Morten Mau-Sorensen
机构
[1] Novartis Pharmaceuticals Corporation,Medical Oncology Department
[2] Fondazione IRCCS-Istituto Nazionale Dei Tumori,Department of Oncology
[3] Hospital Universitario La Paz,undefined
[4] IdiPAZ,undefined
[5] CIOCC-Grupo Hospitalario de Madrid,undefined
[6] Hosp. de Sanchinarro,undefined
[7] Henry Ford Cancer Institute,undefined
[8] Rigshospitalet,undefined
来源
Cancer Chemotherapy and Pharmacology | 2021年 / 87卷
关键词
ALK inhibitor; Ceritinib; Drug–drug interaction; Pharmacokinetics; CYP3A; CYP2C9; Midazolam; Warfarin;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:475 / 486
页数:11
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