Design, synthesis, and antiproliferative activities of novel thiazolyl-pyrazole hybrid derivatives

被引:0
作者
Burak Kuzu
Ali Ergüç
Fuat Karakuş
Ege Arzuk
机构
[1] Van Yüzüncü Yıl University,Department of Pharmaceutical Chemistry, Faculty of Pharmacy
[2] İzmir Kâtip Çelebi University,Department of Pharmaceutical Toxicology, Faculty of Pharmacy
[3] Van Yüzüncü Yıl University,Department of Pharmaceutical Toxicology, Faculty of Pharmacy
[4] Ege University,Department of Pharmaceutical Toxicology, Faculty of Pharmacy
来源
Medicinal Chemistry Research | 2023年 / 32卷
关键词
Thiazolyl-pyrazole; Antiproliferation; ADMET; SAR;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:1690 / 1700
页数:10
相关论文
共 50 条
[31]   Design and Synthesis of C-19 Isosteviol Derivatives as Potent and Highly Selective Antiproliferative Agents [J].
Luan, Tian ;
Cao, Li-Hua ;
Deng, Hao ;
Shen, Qing-Kun ;
Tian, Yu-Shun ;
Quan, Zhe-Shan .
MOLECULES, 2019, 24 (01)
[32]   Design, synthesis, characterization and anti-inflammatory evaluation of novel pyrazole amalgamated flavones [J].
Chavan, Hemant V. ;
Bandgar, Babasaheb P. ;
Adsul, Laxman K. ;
Dhakane, Valmik D. ;
Bhale, Pravin S. ;
Thakare, Vishnu N. ;
Masand, Vijay .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (05) :1315-1321
[33]   Novel Pyrazole Acyl(thio)urea Derivatives Containing a Biphenyl Scaffold as Potential Succinate Dehydrogenase Inhibitors: Design, Synthesis, Fungicidal Activity, and SAR [J].
Sun, Na-Bo ;
Min, Li-Jing ;
Sun, Xin-Peng ;
Zhai, Zhi-Wen ;
Bajsa-Hirschel, Joanna ;
Wei, Zhe-Cheng ;
Hua, Xue-Wen ;
Cantrell, Charles L. ;
Xu, Hao ;
Duke, Stephen O. ;
Liu, Xing-Hai .
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2024, 72 (05) :2512-2525
[34]   Synthesis, characterization and molecular modeling approach of hybrid pyrazole based thiazolidinone derivatives: An estimation and inhibition of diabetes mellitus [J].
Hawsawia, Mohammed B. ;
Khan, Shoaib ;
Iqbal, Tayyiaba ;
Hussain, Rafaqat ;
Khan, Yousaf ;
Zahoor, Tayyaba ;
Dera, Ayed A. .
JOURNAL OF MOLECULAR STRUCTURE, 2025, 1322
[35]   Design and Synthesis of Pyrazole-Substituted 9-Anilinoacridine Derivatives and Evaluation against Breast Cancer [J].
Murugesan, Dhinesh Kumar ;
Rajagopal, Kalirajan ;
Vijayakumar, Arumugam R. ;
Sundararajan, Gothandam ;
Raman, Kannan ;
Byran, Gowramma ;
Murugesan, Esakkimuthukumar ;
Gupta, Jeetendra Kumar ;
Kankate, Rani S. ;
Nainu, Firzan ;
Barua, Rashu ;
Ahmad, Sheikh F. ;
Bin Emran, Talha .
JOURNAL OF BIOLOGICAL REGULATORS AND HOMEOSTATIC AGENTS, 2024, 38 (04) :2845-2859
[36]   Design, synthesis, biological and in silico evaluation of coumarin-hydrazone derivatives as tubulin targeted antiproliferative agents [J].
Pilli, Govindaiah ;
Dumala, Naresh ;
Mattan, Irshad ;
Grover, Paramjit ;
Prakash, Jaya M. .
BIOORGANIC CHEMISTRY, 2019, 91
[37]   Design, synthesis and structure-activity relationships of antiproliferative 1,3-disubstituted urea derivatives [J].
Li, Huan-Qiu ;
Zhu, Tao-Tao ;
Yan, Tao ;
Luo, Yin ;
Zhu, Hai-Liang .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2009, 44 (02) :453-459
[38]   Design, Synthesis, and Biological Activity of Novel Diazabicyclo Derivatives as Safeners [J].
Zhang, Yuan-Yuan ;
Gao, Shuang ;
Liu, Yong-Xuan ;
Wang, Chen ;
Jiang, Wei ;
Zhao, Li-Xia ;
Fu, Ying ;
Ye, Fei .
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2020, 68 (11) :3403-3414
[39]   Studies on the Synthesis and Biological Activities of Novel Dihydroquinazolinone-Containing Caffeine Derivatives [J].
Wang Lei ;
Yu Shujing ;
Yang N ;
Wang Baolei .
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 43 (01) :299-307
[40]   Design, Synthesis, Insecticidal Activity, and SAR of Aryl Isoxazoline Derivatives Containing Pyrazole-5-carboxamide Motif [J].
Zhong, Liang-Kun ;
Sun, Xin-Peng ;
Han, Liang ;
Tan, Cheng-Xia ;
Weng, Jian-Quan ;
Xu, Tian-Ming ;
Shi, Jian-Jun ;
Liu, Xing-Hai .
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 71 (40) :14458-14470