Synthesis of 7-aminopyrazolo[3,4-c]pyridine as a probe for the preparation of compounds of pharmacological interest

被引：0
|
作者：
Kourafalos, VN
Marakos, P
Pouli, N
Terzis, A
Townsend, LB
机构：
[1] Univ Athens, Dept Pharm, Div Pharmaceut Chem, GR-15771 Athens, Greece
[2] NCSR Demokritos, Inst Sci Mat, GR-15310 Athens, Greece
[3] Univ Michigan, Coll Pharm, Dept Med Chem, Ann Arbor, MI 48109 USA
[4] Univ Michigan, Coll Literature Sci & Arts, Dept Chem, Ann Arbor, MI 48109 USA
来源：
HETEROCYCLES | 2002年 / 57卷 / 12期
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D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A synthetic route towards the preparation of 7-aminopyrazolo[3,4-c]pyridine is developed, starting from the readily accessible 2-amino-4-methyl-3-nitropyridine. The unexpected formation of 7-methylimidazolo[4,5-b]pyridin-2-one during the reaction sequence is also described.
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页码：2335 / 2343
页数：9
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