A conventional route for the synthesis of new oxazolidin-2-one derivatives with β-aminoalanines

被引：9
作者：
Fujisaki, F [1 ]
Abe, N [1 ]
Sumoto, K [1 ]
机构：
[1] Fukuoka Univ, Fac Pharmaceut Sci, Jonan Ku, Fukuoka 8140180, Japan
来源：
CHEMICAL & PHARMACEUTICAL BULLETIN | 2004年 / 52卷 / 10期
关键词：
oxazolidin-2-one; oxazolidinone; beta-aminoalanine; cyclization; benzoylation; dehydration;
D O I：
10.1248/cpb.52.1238
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A conventional new route to the novel oxazolidin-2-one derivatives (3a-f) having two substituents on N-3 and C-4 in the oxazolidin-2-one ring was established with racemic beta-aminoalanine derivatives (1) as the key starting materials.
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收藏
页码：1238 / 1241
页数：4
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