Preliminary results from a phase 1/2 study of INCB054828, a highly selective fibroblast growth factor receptor (FGFR) inhibitor, in patients with advanced malignancies

被引:8
作者
Saleh, Mansoor
Gutierrez, Martin E.
Subbiah, Vivek
Smith, David C.
Asatiani, Ekaterine
Lihou, Christine F.
Zhen, Huiling
Yeleswaram, Swamy
Ji, Tao
Nemunaitis, John
机构
关键词
D O I
10.1158/1538-7445.AM2017-CT111
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
CT111
引用
收藏
页数:2
相关论文
共 50 条
[41]   Tinengotinib, a novel fibroblast growth factor receptor (FGFR) inhibitor, is potent against resistance mutations in FGFR1/2/3 [J].
Qiang, Xiaoyan ;
Yu, Qi ;
Fan, Jean ;
Wu, Frank ;
Sun, Caixia ;
Peng, Peng .
CANCER RESEARCH, 2023, 83 (08)
[42]   Phase I study of the irreversible fibroblast growth factor receptor 1-4 inhibitor futibatinib in Japanese patients with advanced solid tumors [J].
Doi, Toshihiko ;
Shitara, Kohei ;
Kojima, Takashi ;
Kuboki, Yasutoshi ;
Matsubara, Nobuaki ;
Bando, Hideaki ;
Yoh, Kiyotaka ;
Naito, Yoichi ;
Hirai, Hiroshi ;
Kurokawa, Yukinori ;
Kato, Terufumi ;
Morizane, Chigusa .
CANCER SCIENCE, 2023, 114 (02) :574-585
[43]   Discovery of BW710 as a potent, selective and orally bioavailable fibroblast growth factor receptor 2 (FGFR2) inhibitor [J].
Yang, Bowen ;
Xun, Qiuju ;
Tian, Yuan ;
Li, Huiqiong ;
Wu, Pinglian ;
Zhou, Yang ;
Chang, Shaohua ;
Wang, Zhen ;
Ding, Ke ;
Ma, Dawei .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 287
[44]   Phase I study of fibroblast growth factor receptor 2 antibody-drug conjugate (FGFR2-ADC) BAY 1187982 in patients with advanced cancer [J].
Kim, Sung-Bae ;
Meric-Bernstam, Funda ;
Berlin, Jordan ;
Wittemer-Rump, Sabine ;
Osada, Motonobu ;
Valencia, Ray ;
Babich, Aleksei ;
Liu, Rong ;
Hwang, Andy ;
Tanigawa, Takahiko ;
Reetz, Frank ;
Laurent, Dirk ;
Kalyan, Aparna .
CANCER RESEARCH, 2017, 77
[45]   A Phase 2 Study of Erdafitinib in Patients with Advanced Solid Tumors and Fibroblast Growth Factor Receptor Gene Alterations [J].
Pant, S. ;
Tabernero, J. ;
Massard, C. ;
Hyman, D. M. ;
Witt, O. ;
Doi, T. ;
Qin, S. ;
Lu-Emerson, C. ;
Hargrave, D. ;
Garcia-Corbacho, J. ;
Little, S. ;
Tolbert, J. ;
Santiago-Walker, A. ;
Moy, C. ;
Hammond, C. ;
Lau, Y. Y. ;
Sweiti, H. ;
Schuler, M. .
JOURNAL OF THORACIC ONCOLOGY, 2021, 16 (03) :S673-S673
[46]   First-in-human phase I study of E7090, a novel selective fibroblast growth factor receptor inhibitor, in patients with advanced solid tumors [J].
Koyama, Takafumi ;
Shimizu, Toshio ;
Iwasa, Satoru ;
Fujiwara, Yutaka ;
Kondo, Shunsuke ;
Kitano, Shigehisa ;
Yonemori, Kan ;
Shimomura, Akihiko ;
Iizumi, Sakura ;
Sasaki, Tatsuya ;
Furuse, Junji ;
Yamamoto, Noboru .
CANCER SCIENCE, 2020, 111 (02) :571-579
[47]   A novel mRNA-based patient selection strategy identifies fibroblast growth factor receptor (FGFR) inhibitor-sensitive tumors: Results from rogaratinib Phase-1 study [J].
Joerger, M. ;
Soo, R. A. ;
Cho, B. C. ;
Navarro, A. ;
Sayehli, C. M. ;
Richly, H. ;
Tai, D. ;
Kim, D-W. ;
Wolf, J. ;
Cassier, P. ;
Bender, S. ;
Ellinghaus, P. ;
Ince, S. ;
Rajagopalan, P. ;
Ocker, M. ;
Schuler, M. .
ANNALS OF ONCOLOGY, 2017, 28
[48]   Preliminary results from fight-102: a phase 1 study of pemigatinib in Japanese patients with advanced malignancies [J].
Kuboki, Yasutoshi ;
Furukawa, Masayuki ;
Takahashi, Yasuo ;
Mizuno, Nobumasa ;
Hara, Hiroki ;
Ueno, Makoto ;
Ioka, Tatsuya ;
Takahashi, Shunji ;
Shimizu, Toshio ;
Lihou, Christine F. ;
Tian, Chenwei ;
Ji, Tao ;
Fujiwara, Yutaka .
ANNALS OF ONCOLOGY, 2019, 30
[49]   A Phase 2 Study of Futibatinib (TAS-120) in Patients with Myeloid or Lymphoid Neoplasms Harboring Fibroblast Growth Factor Receptor (FGFR) 1 Rearrangements [J].
Kiladjian, Jean-Jacques ;
Shitara, Kohei ;
Rosen, Lee Stephen ;
Rha, Sun Young ;
He, Aiwu ;
Oh, Do-Youn ;
Melisi, Davide ;
Iwasa, Satoru ;
Jiang, Yixing ;
Liu, Sherry ;
Takahashi, Osamu ;
Ribrag, Vincent .
BLOOD, 2021, 138 :3656-+
[50]   FIGHT-207: Phase 2 study of pemigatinib in patients with previously treated, locally advanced/metastatic or unresectable solid tumor malignancies harboring activating fibroblast growth factor receptor (FGFR) gene alterations [J].
Feliz, Luis ;
Asatiani, Ekaterine ;
Lihou, Christine ;
Zhen, Huiling ;
Silverman, Ian ;
Ahnert, Jordi Rodon .
MOLECULAR CANCER THERAPEUTICS, 2019, 18 (12)