1-aza sugars, apparent transition state analogues of equatorial glycoside formation/cleavage

被引：306
作者：
Bols, M [1 ]
机构：
[1] Aarhus Univ, Dept Chem, DK-8000 Aarhus C, Denmark
来源：
ACCOUNTS OF CHEMICAL RESEARCH | 1998年 / 31卷 / 01期
关键词：
D O I：
10.1021/ar970058r
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
[No abstract available]
引用
收藏
页码：1 / 8
页数：8
相关论文
共 60 条
  • [1] 7-carbon mimics of D-glucose and L-fucose: Activation by 6R-, and inactivation by 6S, -6C-methylglucose of glycogen synthase: Inhibition of glucokinase and/or glucose-6-phosphatase
    Bleriot, Y
    Smelt, KH
    Cadefau, J
    Bollen, M
    Stalmans, W
    Biggadike, K
    Johnson, LN
    Oikonomakos, NG
    Lane, AL
    Crook, S
    Watkin, DJ
    Fleet, GWJ
    [J]. TETRAHEDRON LETTERS, 1996, 37 (39) : 7155 - 7158
  • [2] Synthesis of a ribofuranosyl cation mimic
    Bols, M
    [J]. TETRAHEDRON LETTERS, 1996, 37 (12) : 2097 - 2100
  • [3] 1-azafagomine: A hydroxyhexahydropyridazine that potently inhibits enzymatic glycoside cleavage
    Bols, M
    Hazell, RG
    Thomsen, IB
    [J]. CHEMISTRY-A EUROPEAN JOURNAL, 1997, 3 (06) : 940 - 947
  • [4] Bols M., 1995, CARBOHYDRATE BUILDIN
  • [5] GUANIDINE ANALOGS OF A DEOXYSUGAR
    CHAN, AWY
    GANEM, B
    [J]. TETRAHEDRON LETTERS, 1995, 36 (06) : 811 - 814
  • [6] AN IMINO-LINKED CARBA-DISACCHARIDE ALPHA-DEUTERIUM-MANNOSIDASE INHIBITOR
    COTTAZ, S
    BRIMACOMBE, JS
    FERGUSON, MAJ
    [J]. CARBOHYDRATE RESEARCH, 1993, 247 : 341 - 345
  • [7] REVERSIBLE INHIBITORS OF BETA-GLUCOSIDASE
    DALE, MP
    ENSLEY, HE
    KERN, K
    SASTRY, KAR
    BYERS, LD
    [J]. BIOCHEMISTRY, 1985, 24 (14) : 3530 - 3539
  • [8] DESLONGCHAMPS P, 1983, STEREOELECTRONIC EFF, P31
  • [9] Evaluation of isofagomine and its derivatives as potent glycosidase inhibitors
    Dong, WL
    Jespersen, T
    Bols, M
    Skrydstrup, T
    Sierks, MR
    [J]. BIOCHEMISTRY, 1996, 35 (08) : 2788 - 2795
  • [10] CONFIGURATIONALLY SELECTIVE TRANSITION-STATE ANALOG INHIBITORS OF GLYCOSIDASES - A STUDY WITH NOJIRITETRAZOLES, A NEW CLASS OF GLYCOSIDASE INHIBITORS
    ERMERT, P
    VASELLA, A
    WEBER, M
    RUPITZ, K
    WITHERS, SG
    [J]. CARBOHYDRATE RESEARCH, 1993, 250 (01) : 113 - 128
123456