Progress in Synthesis of 2-Substituted Benzothiazole Compounds

被引：6
|
作者：
Zhang, Jun [1 ]
Liu, Yafei [1 ]
Zhang, Yurong [1 ]
Hu, Liang [1 ]
Han, Shiqing [1 ]
机构：
[1] Nanjing Tech Univ, Coll Biotechnol & Pharmaceut Engn, Nanjing 211816, Peoples R China
来源：
CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2021年 / 41卷 / 03期
关键词：
2-substituted benzothiazole; condensation; dehydrogenation; redox; arylation; coupling cyclization; ONE-POT SYNTHESIS; COPPER-CATALYZED SYNTHESIS; REDOX CYCLIZATION REACTION; S BOND FORMATION; C-H ARYLATION; ELEMENTAL SULFUR; N-HETEROCYCLES; ACCEPTORLESS DEHYDROGENATION; O-CHLORONITROBENZENES; SUBSTITUTED ANILINES;
D O I：
10.6023/cjoc202007036
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The application and research of 2-substituted benzothiazoles in biomedicine, materials science and other fields have made their synthetic methods widely concerned. Based on the research of traditional synthetic methods, the development of new methods such as elemental sulfur-mediated redox reaction and dehydroaromatization of saturated compounds could provide more possibilities for the synthesis of benzothiazole derivatives. In addition, the application of new metal-organic framework catalysts, combined ionic liquids/gels, ultrasound and microwave assist in recent years have greatly enriched the synthesis of benzothiazole derivatives. The synthetic method of 2-substituted benzothiazoles in recent years is analyzed.
引用
收藏
页码：1053 / 1071
页数：19
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