Synthesis of pyrimidine-annelated heterocycles:: Regioselective synthesis of 1,3,6-trialkyl thieno[3,2-d]-pyrimidine-2,4-diones

被引：9

作者：

Majumdar, KC ^{[1
]}

Jana, NK ^{[1
]}

机构：

[1] Univ Kalyani, Dept Chem, Kalyani 741235, W Bengal, India

来源：

SYNTHETIC COMMUNICATIONS | 2000年 / 30卷 / 22期

关键词：

D O I：

10.1080/00397910008087036

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Thermal [3,3] sigmatropic rearrangement of a number of 1,3-dimethyl-5-(prop-2-ynylthio)uracils (4a-j) afforded the title compounds 5a-j in 60-82% yields.

引用

页码：4183 / 4196

页数：14

共 50 条

[21] Convenient synthesis of 3-(1-carboxyalkyl)pyrido-[2,3-d]pyrimidine-2,4-diones
Saoud M.
Benabdelouahab F.B.
Guemmout F.E.
Romerosa A.
Chemistry of Heterocyclic Compounds, 2002, 38 (03) : 306 - 309
[22] SYNTHESIS OF NEW 1H,3H-PYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES
BRUNEL, S
MONTGINOUL, C
TORREILLES, E
GIRAL, L
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1980, 17 (02) : 235 - 240
[23] SYNTHESIS OF 8-METHYL-1,2,3,4-TETRAHYDROPYRIDO-[3,4-D]PYRIMIDINE-2,4-DIONES
KUJUNDZIC, N
GLUNCIC, B
CROATICA CHEMICA ACTA, 1991, 64 (04) : 599 - 606
[24] Synthesis and evaluation of thieno[3,2-d]pyrimidine derivatives as novel FMS inhibitors
Kim, Yu-Yon
Choi, Jaeyul
Choi, Kyungjin
Park, Changhee
Kim, Young Hoon
Suh, Kwee Hyun
Ham, Young Jin
Jang, Sun Young
Lee, Kyu-Hang
Hwang, Kwang Woo
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (02) : 271 - 275
[25] SYNTHESIS OF SOME NOVEL THIENO[3,2-d]PYRIMIDINE DERIVATIVES OF PHARMACEUTICAL INTEREST
Refat, Hala M.
Fadda, Ahmed A.
El-Mekawy, Rasha E.
Sleat, Aliaa M.
HETEROCYCLES, 2015, 91 (12) : 2271 - 2284
[26] Synthesis and anti-HIV-1 evaluation of 1,5-disubstituted pyrimidine-2,4-diones
Loksha, Yasser M.
Globisch, Daniel
Pedersen, Erik B.
La Colla, Paolo
Collu, Gabriella
Loddo, Roberta
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2008, 45 (04) : 1161 - 1166
[27] A FACILE SYNTHESIS OF 7-SUBSTITUTED PYRIMIDO[4,5-D]-PYRIMIDINE-2,4-DIONES
HIROTA, K
KITADE, Y
SAJIKI, H
MAKI, Y
SYNTHESIS-STUTTGART, 1984, (07): : 589 - 590
[28] Convenient One-Pot Synthesis of Functionalized Thieno[3,2-d]pyrimidine and Thieno[2,3-d]pyrimidine Derivatives
Fernandez-Mato, Antonio
Peinador, Carlos
Maria Quintela, Jose
SYNTHESIS-STUTTGART, 2011, (20): : 3323 - 3331
[29] Regioselective synthesis of 6H-pyrano[3,2-e]pyrimidine-2,4-dione
Majumdar, KC
Das, U
SYNTHETIC COMMUNICATIONS, 1997, 27 (22) : 4013 - 4019
[30] SYNTHESIS AND ANTIVIRAL STUDY OF CYCLOPENTANO[D]PYRIMIDINE-2,4-DIONES AND OCTAHYDROQUINAZOLINE-2,4-DIONES ACYCLIC NUCLEOSIDES AS POTENTIAL ANTI-HIV AGENTS
RENAULT, J
LADUREE, D
ROBBA, M
NUCLEOSIDES & NUCLEOTIDES, 1994, 13 (04): : 891 - 901

← 1 2 3 4 5 →