A concise synthesis of (S)-(-)-3-(2-carboxy-4-pyrrolyl)-alanine

被引：18
作者：
Adamczyk, M [1 ]
Johnson, DD [1 ]
Reddy, RE [1 ]
机构：
[1] Abbott Labs, Div Diagnost, Dept Chem, Abbott Pk, IL 60064 USA
来源：
TETRAHEDRON-ASYMMETRY | 2000年 / 11卷 / 15期
关键词：
D O I：
10.1016/S0957-4166(00)00266-4
中图分类号：
O61 [无机化学];
学科分类号：
070301 ; 081704 ;
摘要：
A convergent synthesis of (S)-(-)-3-(2-carboxy-4-pyrrolyl)-alanine (CPA) 1, a non-proteinogenic amino acid is described starting from a commercially available dimethyl L-aspartate 2 in good overall yield. (C) 2000 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：3063 / 3068
页数：6
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