Antifeedant activity of some pentacyclic triterpene acids and their fatty acid ester analogues

被引:52
作者
Mallavadhani, UV [1 ]
Mahapatra, A
Raja, SS
Manjula, C
机构
[1] CSIR, Reg Res Lab, Forest & Marine Prod Dept, Nat Resources Div, Bhubaneswar 751013, Orissa, India
[2] Osmania Univ, Dept Zool, Hyderabad 500017, Andhra Pradesh, India
关键词
antifeedant activity; ursolic acid; oleanolic acid; fatty acid esters; tobacco caterpillar; Spodoptera litura;
D O I
10.1021/jf020691d
中图分类号
S [农业科学];
学科分类号
09 ;
摘要
The 3-O-fatty acid ester derivatives (C-12-C-18) of two pentacyclic triterpenic acids, ursolic acid and oleanolic acid, were synthesized under mild esterification conditions in excellent yields (80-85%) and screened for their antifeedant activity, together with the parent acids, against the agricultural pest tobacco caterpillar larvae (Spodoptera litura F) in a no-choice laboratory study. The Urs-12-ene-28-carboxy-3beta- octadecanoate and olean-12-ene-28-carboxy-3beta-hexadecanoate were found to exhibit exceptionally potent antifeedant activities at 50 mug/cm(2) concentration, even after 48 h.
引用
收藏
页码:1952 / 1955
页数:4
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