2-chloro-4,6-dimethoxy-1,3,5-triazine: A new effective and convenient coupling reagent for cephalosporin derivatives

被引：13
|
作者：
Lee, HW [1 ]
Kang, TW [1 ]
Cha, KH [1 ]
Kim, EN [1 ]
Choi, NH [1 ]
Kim, JW [1 ]
Hong, CI [1 ]
机构：
[1] Chong Kun Dang Corp, Res Inst, Seoul 152600, South Korea
来源：
SYNTHETIC COMMUNICATIONS | 1998年 / 28卷 / 08期
关键词：
D O I：
10.1080/00397919808006831
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Chloro-4,6-dimethoxy-1,3,5-triazine(CDMT) 2 was reacted with 2-(2-amino-4-thiazolyl)-2-syn-alkoxyiminoacetic acid 1 to give an active ester intermediate 3.
引用
收藏
页码：1339 / 1349
页数：11
相关论文
共 50 条
  • [41] DERIVATIVES OF S-TRIAZINE .1. INTERACTION OF 2-CHLORO-4,6-DIMETHOXY-S-TRIAZINE WITH SODIUM MALONIC ESTER
    VAKHATOVA, GM
    ANISIMOVA, OS
    YAKHONTOV, LN
    KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII, 1979, (11): : 1557 - 1560
  • [42] 2-CHLORO-4,6-DIBENZYLOXY-1,3,5-TRIAZINE AND N-(3,5-DIBENZYLOXY-1,3,5-TRIAZINYL-1)AMMONIUM TETRAFLUOROBORATES AS NEW, HIGHLY EFFICIENT COUPLING REAGENTS FOR PEPTIDE SYNTHESIS IN SOLUTION
    Jastrzabek, K.
    Blaszczyk, M.
    Glowka, M. L.
    Kolesinska, B.
    Papini, A. M.
    Kaminski, Z. J.
    JOURNAL OF PEPTIDE SCIENCE, 2004, 10 : 147 - 147
  • [43] Benzyl 4,6-dimethoxy-1,3,5-triazinyl carbonate as N-protecting reagent
    Hioki, K
    Fujiwara, M
    Tani, S
    Kunishima, M
    CHEMISTRY LETTERS, 2002, (01) : 66 - 67
  • [44] STRUCTURE OF CONDENSATION PRODUCT OF METHYL CYANOACETATE AND 2,4-DIMETHOXY-6-CHLORO-1,3,5-TRIAZINE
    WEBER, AJM
    HUYSMANS, WGB
    MIJS, WJ
    BOVEE, WMMJ
    SMIDT, J
    VRIEND, J
    RECUEIL DES TRAVAUX CHIMIQUES DES PAYS-BAS-JOURNAL OF THE ROYAL NETHERLANDS CHEMICAL SOCIETY, 1978, 97 (04): : 107 - 110
  • [45] 2-AMINO-4,6-DIAZIDO-1,3,5-TRIAZINE
    HENRY, RA
    JOURNAL OF ORGANIC CHEMISTRY, 1966, 31 (06): : 1973 - &
  • [46] Transformation of Tertiary Amines into Alkylating Reagents by Treatment with 2-Chloro-4,6-dimethoxy-1,3,5-triazine. A Synthetic Application of Side-Reaction Accompanying Coupling by Means of 4-(4,6-Dimethoxy-[1,3,5]triazin-2-yl)-4-methyl-morpholin-4-ium Chloride (DMTMM)
    Kolesinska, B.
    Kaminski, Z. J.
    POLISH JOURNAL OF CHEMISTRY, 2008, 82 (11) : 2115 - 2123
  • [47] STRUCTURES OF 2-CHLORO-4-CYCLOHEXYLAMINO-6-METHOXY-1,3,5-TRIAZINE AND 2-CHLORO-4-METHOXY-6-PIPERIDINO-1,3,5-TRIAZINE
    GLOWKA, ML
    IWANICKA, I
    ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 1991, 47 : 616 - 618
  • [48] Synthesis and antitubercular activity of 4,6-diamino-1,3,5-triazine derivatives
    Yun, Chang-Soo
    Choi, Yun-Hee
    Lee, Sang-Ho
    Lee, Ill-Young
    Kim, Pilho
    Park, Tae-Ho
    Oh, Taegwon
    Cho, Sang-Nae
    Camacho, Luis R.
    Beer, David
    Patel, Viral
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 237
  • [49] 2-Chloro-4,6-bis-(2,2,2-trifluoroethoxy)-1,3,5-triazine and N-4,6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2yl)ammonium tetrafluoroborates as highly efficient coupling reagents
    Jastrzabek, Konrad
    Kolesinska, Beata
    Kaminski, Zbigniew J.
    JOURNAL OF PEPTIDE SCIENCE, 2008, 14 (08) : 72 - 72
  • [50] Thermal decomposition of 2,4-diazido-6-trinitromethyl-1,3,5-triazine, 2,4-dimethoxy-6-trinitromethyl-1,3,5-triazine, and 2,4-diazido-6-methoxy-1,3,5-triazine
    V. V. Nedel’ko
    V. V. Zakharov
    B. L. Korsounskii
    T. S. Larikova
    N. V. Chukanov
    A. V. Shastin
    Russian Journal of Physical Chemistry B, 2015, 9 : 885 - 889
12345