2-chloro-4,6-dimethoxy-1,3,5-triazine: A new effective and convenient coupling reagent for cephalosporin derivatives

被引：13
|
作者：
Lee, HW [1 ]
Kang, TW [1 ]
Cha, KH [1 ]
Kim, EN [1 ]
Choi, NH [1 ]
Kim, JW [1 ]
Hong, CI [1 ]
机构：
[1] Chong Kun Dang Corp, Res Inst, Seoul 152600, South Korea
来源：
SYNTHETIC COMMUNICATIONS | 1998年 / 28卷 / 08期
关键词：
D O I：
10.1080/00397919808006831
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Chloro-4,6-dimethoxy-1,3,5-triazine(CDMT) 2 was reacted with 2-(2-amino-4-thiazolyl)-2-syn-alkoxyiminoacetic acid 1 to give an active ester intermediate 3.
引用
收藏
页码：1339 / 1349
页数：11
相关论文
共 50 条
  • [21] Activation of N-benzoyl-2-substituted-2-hydroxymethyl-2-amino acids with chiral coupling reagents prepared in situ from 2-chloro-4,6-dimethoxy-1,3,5-triazine
    Kolesinska, B.
    Kaminska, J. E.
    Miyazawa, T.
    Kaminski, Z. J.
    POLISH JOURNAL OF CHEMISTRY, 2006, 80 (11) : 1817 - 1824
  • [22] On the electroreduction mechanism of 2-chloro-4,6-diamino-1,3,5-triazine on mercury electrodes
    Pérez, R
    Galvín, RM
    Mellado, JMR
    Montoya, MR
    JOURNAL OF THE ELECTROCHEMICAL SOCIETY, 2003, 150 (08) : E389 - E395
  • [23] 2-Chloro-4,6-bis(piperidin-1-yl)-1,3,5-triazine
    Vennila, Jasmine P.
    Thiruvadigal, D. John
    Kavitha, Helen P.
    Chakkaravarthi, G.
    Manivannan, V.
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2011, 67 : O312 - U150
  • [24] PERHYDROLYSIS OF 2-CHLORO-4,6-DIMETHOXY-S-TRIAZINE
    SPEAKMAN, PRH
    CHEMISTRY & INDUSTRY, 1977, (06) : 232 - 232
  • [25] PREDICTION OF ACYLATION CAPABILITY OF S-TRIAZINYL (ACTIVE) ESTERS BASED ON STRUCTURES OF APPROPRIATE ETHERS - CRYSTAL-STRUCTURES OF 2 2-ARYLOXY-4,6-DIMETHOXY-1,3,5-TRIAZINES - 2-(2-ETHOXYCARBONYLPHENOXY)-4,6-DIMETHOXY-1,3,5-TRIAZINE AND 2-(4-METHYLPHENOXY)-4,6-DIMETHOXY-1,3,5-TRIAZINE
    GLOWKA, ML
    KAMINSKI, ZJ
    SOBANSKA, AW
    POLISH JOURNAL OF CHEMISTRY, 1994, 68 (09) : 1731 - 1741
  • [26] An Efficient One-pot N-Acylation of Deoxy- and Ribo-cytidine Using Carboxylic Acids Activated in situ with 2-Chloro-4,6-dimethoxy-1,3,5-triazine
    Rode, Ambadas B.
    Son, Sang Jun
    Hong, In Seok
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2010, 31 (07) : 2061 - 2064
  • [27] A convenient method for the conversion of a carboxy group into a 4,6-dimethoxy-1,3,5-triazine group:: Application to N-benzylpyroglutamic acids
    Oudir, Souhila
    Rigo, Benoit
    Henichart, Jean-Pierre
    Gautret, Philippe
    SYNTHESIS-STUTTGART, 2006, (17): : 2845 - 2848
  • [28] Fluorous coupling reagents: Application of 2-chloro-4,6-bis[(heptadecafluorononyl)oxy]-1,3,5-triazine in peptide synthesis
    Markowicz, MW
    Dembinski, R
    SYNTHESIS-STUTTGART, 2004, (01): : 80 - 86
  • [29] Derivatives of 2,4-dimethoxy-1,3,5-triazine
    Fridman, N
    Kapon, M
    Kaftory, M
    ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 2003, 59 : O687 - O689
  • [30] Diazo-Transfer Reagent 2-Azido-4,6-dimethoxy-1,3,5-triazine Displays Highly Exothermic Decomposition Comparable to Tosyl Azide
    Green, Sebastian P.
    Payne, Andrew D.
    Wheelhouse, Katherine M.
    Hallett, Jason P.
    Miller, Philip W.
    Bull, James A.
    JOURNAL OF ORGANIC CHEMISTRY, 2019, 84 (09): : 5893 - 5898
12345