Design, Synthesis and Biological Activities of Novel Dual-Chiral Carbon and Sulfur Pyridine Phthalic Acid Diamide Derivatives

被引：6

作者：

Meng, Xiangde ^{[1
]}

Zhou, Sha ^{[1
]}

Xie, Yongtao ^{[1
]}

Zhao, Yu ^{[1
]}

Xiong, Lixia ^{[1
]}

Zhou, Sha ^{[1
]}

Li, Zhengming ^{[1
]}

机构：

[1] Nankai Univ, Inst Elementoorgan Chem, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2017年 / 37卷 / 04期

基金：

中国国家自然科学基金;

关键词：

pyridine; phthalic acid diamides; synthesis; insecticidal activity; dual-chiral; INSECTICIDAL ACTIVITIES; SULFILIMINYL;

D O I：

10.6023/cjoc201610027

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

In order to find efficient, low toxicity, eco-friendly insecticides, novel chiral carbon and sulfur phthalic acid diamide derivatives containing pyridine substitute were designed and synthesized for further studying the structure-activity relationship of dual-chiral sulfilimines and sulfoximines. Their structures were confirmed by NMR and HRMS. The preliminary results of biological evaluation showed that the most compounds exhibited moderate larvicidal activity. These results provide a theoretical basis for the study of the dicarboxamide structures containing sulfiliminyl and sulfoximinyl moieties.

引用

页码：908 / 913

页数：6

共 20 条

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