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VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications
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JOURNAL OF MEDICINAL CHEMISTRY,
2023, 66 (18)
:13148-13171

Castellani, Beatrice
论文数: 0 引用数: 0
h-index: 0
机构:
Mol Horizon Srl, I-06084 Bettona, Italy Univ Perugia, Dept Chem Biol & Biotechnol, I-06123 Perugia, Italy

论文数: 引用数:
h-index:
机构:

Di Bona, Stefano
论文数: 0 引用数: 0
h-index: 0
机构:
Mol Horizon Srl, I-06084 Bettona, Italy Univ Perugia, Dept Chem Biol & Biotechnol, I-06123 Perugia, Italy

论文数: 引用数:
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Desantis, Jenny
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Chem Biol & Biotechnol, I-06123 Perugia, Italy Univ Perugia, Dept Chem Biol & Biotechnol, I-06123 Perugia, Italy

Goracci, Laura
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h-index: 0
机构:
Univ Perugia, Dept Chem Biol & Biotechnol, I-06123 Perugia, Italy Univ Perugia, Dept Chem Biol & Biotechnol, I-06123 Perugia, Italy
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Designed, synthesized and biological evaluation of proteolysis targeting chimeras (PROTACs) as AR degraders for prostate cancer treatment
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Liang, Jian-Jia
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Xie, Hang
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Yang, Rui-Hua
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Wang, Ni
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Zheng, Zi-Jun
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Zhou, Chen
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Wang, Ya-Lei
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Wang, Zhi-Jia
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Liu, Hong-Min
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Shan, Li-Hong
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Ke, Yu
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BIOORGANIC & MEDICINAL CHEMISTRY,
2021, 45

Liang, Jian-Jia
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h-index: 0
机构:
Wuhan Univ, Sch Pharm, Wuhan 430072, Hubei, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Xie, Hang
论文数: 0 引用数: 0
h-index: 0
机构:
Fudan Univ, Sch Pharm, Shanghai 201203, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Yang, Rui-Hua
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h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Wang, Ni
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Zheng, Zi-Jun
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Zhou, Chen
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h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Wang, Ya-Lei
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Wang, Zhi-Jia
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Liu, Hong-Min
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Shan, Li-Hong
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China

Ke, Yu
论文数: 0 引用数: 0
h-index: 0
机构:
Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
Collaborat Innovat Ctr New Drug Res & Safety Eval, Zhengzhou 450001, Henan, Peoples R China
Minist Educ China, Key Lab Adv Drug Preparat Technol, Beijing, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Henan, Peoples R China
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Targeting Oncoproteins for Degradation by Small Molecule-Based Proteolysis-Targeting Chimeras (PROTACs) in Sex Hormone-Dependent Cancers
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Liu, Li
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Shi, Lihong
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Wang, Zhaodi
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Zeng, Jun
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Wang, Yue
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Xiao, Hongtao
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Zhu, Yongxia
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FRONTIERS IN ENDOCRINOLOGY,
2022, 13

Liu, Li
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China
Southwest Med Univ, Dept Dermatol, Affiliated Hosp, Luzhou, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China

Shi, Lihong
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China

Wang, Zhaodi
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h-index: 0
机构:
Henan Univ, Henan Prov Peoples Hosp, Dept Gynecol, Peoples Hosp, Zhengzhou, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China

Zeng, Jun
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China

Wang, Yue
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h-index: 0
机构:
Henan Univ, Henan Prov Peoples Hosp, Dept Gynecol, Peoples Hosp, Zhengzhou, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China

Xiao, Hongtao
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China

Zhu, Yongxia
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China Univ Elect Sci & Technol China, Sichuan Canc Hosp & Inst, Sichuan Canc Ctr, Sch Med,Dept Clin Pharm, Chengdu, Peoples R China
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Computational methods and key considerations for in silico design of proteolysis targeting chimera (PROTACs)
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INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES,
2024, 277

Abbas, Amr
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h-index: 0
机构:
Zhejiang Sci Tech Univ, Coll Life Sci & Med, Hangzhou 310018, Peoples R China
Cairo Univ, Fac Pharm, Pharmaceut Chem Dept, Cairo 11562, Egypt Zhejiang Sci Tech Univ, Coll Life Sci & Med, Hangzhou 310018, Peoples R China

Ye, Fei
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h-index: 0
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Zhejiang Sci Tech Univ, Coll Life Sci & Med, Hangzhou 310018, Peoples R China Zhejiang Sci Tech Univ, Coll Life Sci & Med, Hangzhou 310018, Peoples R China
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Design, Synthesis and Biological Evaluation of α-Synuclein Proteolysis-Targeting Chimeras
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Wen, Tianzhi
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Chen, Jian
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Zhang, Wenqian
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MOLECULES,
2023, 28 (11)

Wen, Tianzhi
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h-index: 0
机构:
Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China

Chen, Jian
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h-index: 0
机构:
Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China

Zhang, Wenqian
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h-index: 0
机构:
Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China

Pang, Jiyan
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h-index: 0
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Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Chem, Guangzhou 510006, Peoples R China
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Aptamer Proteolysis-Targeting Chimeras (PROTACs): A Novel Strategy to Combat Drug Resistance in Estrogen Receptor α-Positive Breast Cancer
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Feng, Ying
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Zhang, Zhilin
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Guo, Hui
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Tan, Chunyan
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Xu, Naihan
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Tan, Ying
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Jiang, Yuyang
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ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE,
2024, 7 (12)
:3945-3954

Feng, Ying
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h-index: 0
机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Zhang, Zhilin
论文数: 0 引用数: 0
h-index: 0
机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Zhang, Haowei
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h-index: 0
机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Guo, Hui
论文数: 0 引用数: 0
h-index: 0
机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Tan, Chunyan
论文数: 0 引用数: 0
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机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Xu, Naihan
论文数: 0 引用数: 0
h-index: 0
机构:
Shenzhen Polytech Univ, Sch Food & Drug, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Tan, Ying
论文数: 0 引用数: 0
h-index: 0
机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China

Jiang, Yuyang
论文数: 0 引用数: 0
h-index: 0
机构:
Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China Tsinghua Univ, Inst Biopharmaceut & Hlth Engn, Shenzhen Int Grad Sch, State Key Lab Chem Oncogen, Shenzhen 518055, Peoples R China
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Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity
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Darwish, Salma
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Heimburg, Tino
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Herp, Daniel
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Ridinger, Johannes
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Robaa, Dina
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Schmidtkunz, Karin
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Erdmann, Frank
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Schmidt, Matthias
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Romier, Christophe
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Jung, Manfred
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Oehme, Ina
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Sippl, Wolfgang
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INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES,
2022, 23 (14)

Darwish, Salma
论文数: 0 引用数: 0
h-index: 0
机构:
Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany
Alexandria Univ, Fac Pharm, Dept Pharmaceut Chem, Alexandria 21521, Egypt Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

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Heimburg, Tino
论文数: 0 引用数: 0
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机构:
Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Herp, Daniel
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Freiburg, Inst Pharmaceut Sci, D-79104 Freiburg, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Zeyen, Patrik
论文数: 0 引用数: 0
h-index: 0
机构:
Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Salem-Altintas, Rabia
论文数: 0 引用数: 0
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机构:
Hopp Childrens Canc Ctr Heidelberg KiTZ, Neuenheimer Feld 280, D-69120 Heidelberg, Germany
German Canc Res Ctr, Clin Cooperat Unit Pediat Oncol, D-69120 Heidelberg, Germany
German Canc Consortium DKTK, D-69120 Heidelberg, Germany
Heidelberg Univ, Fac Med, D-69120 Heidelberg, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Ridinger, Johannes
论文数: 0 引用数: 0
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机构:
Hopp Childrens Canc Ctr Heidelberg KiTZ, Neuenheimer Feld 280, D-69120 Heidelberg, Germany
German Canc Res Ctr, Clin Cooperat Unit Pediat Oncol, D-69120 Heidelberg, Germany
German Canc Consortium DKTK, D-69120 Heidelberg, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Robaa, Dina
论文数: 0 引用数: 0
h-index: 0
机构:
Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Schmidtkunz, Karin
论文数: 0 引用数: 0
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机构:
Univ Freiburg, Inst Pharmaceut Sci, D-79104 Freiburg, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Erdmann, Frank
论文数: 0 引用数: 0
h-index: 0
机构:
Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Schmidt, Matthias
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Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

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Jung, Manfred
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Freiburg, Inst Pharmaceut Sci, D-79104 Freiburg, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Oehme, Ina
论文数: 0 引用数: 0
h-index: 0
机构:
Hopp Childrens Canc Ctr Heidelberg KiTZ, Neuenheimer Feld 280, D-69120 Heidelberg, Germany
German Canc Res Ctr, Clin Cooperat Unit Pediat Oncol, D-69120 Heidelberg, Germany
German Canc Consortium DKTK, D-69120 Heidelberg, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany

Sippl, Wolfgang
论文数: 0 引用数: 0
h-index: 0
机构:
Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany Martin Luther Univ Halle Wittenberg, Inst Pharm, Dept Med Chem, D-06120 Halle, Saale, Germany
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Identification and Characterization of Von Hippel-Lindau-Recruiting Proteolysis Targeting Chimeras (PROTACs) of TANK-Binding Kinase 1
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Crew, Andrew P.
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Qian, Yimin
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Wang, Jing
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Vigil, Dominico
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Serebrenik, Yevgeniy V.
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Hamman, Brian D.
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Morgan, Alicia
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Ferraro, Caterina
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Siu, Kam
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Neklesa, Taavi K.
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Winkler, James D.
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Crews, Craig M.
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JOURNAL OF MEDICINAL CHEMISTRY,
2018, 61 (02)
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Crew, Andrew P.
论文数: 0 引用数: 0
h-index: 0
机构:
Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Raina, Kanak
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h-index: 0
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Dong, Hanqing
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h-index: 0
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Qian, Yimin
论文数: 0 引用数: 0
h-index: 0
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Wang, Jing
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h-index: 0
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Vigil, Dominico
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA
Agios Pharmaceut, Cambridge, MA USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Serebrenik, Yevgeniy V.
论文数: 0 引用数: 0
h-index: 0
机构:
Yale Univ, Dept Mol Cell & Dev Biol, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Hamman, Brian D.
论文数: 0 引用数: 0
h-index: 0
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Morgan, Alicia
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Ferraro, Caterina
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h-index: 0
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Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Siu, Kam
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h-index: 0
机构:
Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Neklesa, Taavi K.
论文数: 0 引用数: 0
h-index: 0
机构:
Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Winkler, James D.
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h-index: 0
机构:
Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Coleman, Kevin G.
论文数: 0 引用数: 0
h-index: 0
机构:
Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA

Crews, Craig M.
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h-index: 0
机构:
Yale Univ, Dept Mol Cell & Dev Biol, New Haven, CT 06511 USA
Yale Univ, Dept Chem, 225 Prospect St, New Haven, CT 06511 USA
Yale Univ, Dept Pharmacol, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA
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Proteolysis Targeting Chimeras (PROTACs) based on celastrol induce multiple protein degradation for triple-negative breast cancer treatment
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Gan, Xuelan
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Wang, Fan
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Luo, Jianguo
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Zhao, Yunfei
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Wang, Yan
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Yu, Chao
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Chen, Jun
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EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES,
2024, 192

Gan, Xuelan
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h-index: 0
机构:
Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China

Wang, Fan
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Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China

Luo, Jianguo
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Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China

Zhao, Yunfei
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Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China

Wang, Yan
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Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China

Yu, Chao
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Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China

Chen, Jun
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Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China Chongqing Med Univ, Coll Pharm, Chongqing Pharmacodynam Evaluat Engn Technol Res C, Chongqing Key Lab Pharmaceut Metab Res, 1 Yixueyuan Rd, Chongqing 400016, Peoples R China
[40]
Rational Proteolysis Targeting Chimera Design Driven by Molecular Modeling and Machine Learning
[J].
Tan, Shuoyan
;
Chen, Zhenglu
;
Lu, Ruiqiang
;
Liu, Huanxiang
;
Yao, Xiaojun
.
WILEY INTERDISCIPLINARY REVIEWS-COMPUTATIONAL MOLECULAR SCIENCE,
2025, 15 (02)

Tan, Shuoyan
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Zhejiang Univ, Innovat Ctr Yangtze River Delta, State Key Lab Chinese Med Modernizat, Jiaxing, Peoples R China
Zhejiang Univ, Coll Pharmaceut Sci, Hangzhou, Peoples R China Zhejiang Univ, Innovat Ctr Yangtze River Delta, State Key Lab Chinese Med Modernizat, Jiaxing, Peoples R China

Chen, Zhenglu
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Lanzhou Univ, Sch Pharm, Lanzhou, Peoples R China Zhejiang Univ, Innovat Ctr Yangtze River Delta, State Key Lab Chinese Med Modernizat, Jiaxing, Peoples R China

Lu, Ruiqiang
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Macao Polytech Univ, Fac Appl Sci, Macau, Peoples R China Zhejiang Univ, Innovat Ctr Yangtze River Delta, State Key Lab Chinese Med Modernizat, Jiaxing, Peoples R China

Liu, Huanxiang
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Macao Polytech Univ, Fac Appl Sci, Macau, Peoples R China Zhejiang Univ, Innovat Ctr Yangtze River Delta, State Key Lab Chinese Med Modernizat, Jiaxing, Peoples R China

Yao, Xiaojun
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Macao Polytech Univ, Fac Appl Sci, Macau, Peoples R China Zhejiang Univ, Innovat Ctr Yangtze River Delta, State Key Lab Chinese Med Modernizat, Jiaxing, Peoples R China