The synthesis of azabicyclic heterocycles

被引：5
|
作者：
Darout, Etzer [1 ]
Basak, Arindrajit [1 ]
机构：
[1] Groton Labs, Pfizer Global Res & Dev, Groton, CT 06340 USA
来源：
TETRAHEDRON LETTERS | 2010年 / 51卷 / 22期
关键词：
KETONES;
D O I：
10.1016/j.tetlet.2010.03.123
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient approach to a oxa-azabicyclo[3.2.1] derivatives has been achieved via a double-Mannich reaction of N,N-bis(methoxymethyl)-1-phenylethanamine with symmetrical and unsymmetrical ketones. (C) 2010 Elsevier Ltd. All rights reserved.
引用
收藏
页码：2998 / 3001
页数：4
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