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- [1] The PI3K inhibitor, taselisib, has enhanced potency in PIK3CA mutant models through a unique mechanism of actionCANCER RESEARCH, 2017, 77Friedman, L. S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAEdgar, K. A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASong, K.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASchmidt, S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAKirkpatrick, D. S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAPhu, L.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USANannini, M. A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHong, R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USACheng, E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USACrocker, L.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAYoung, A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASampath, D.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [2] The PI3K inhibitor, taselisib (GDC-0032), has enhanced potency in PIK3CA mutant models through a unique mechanism of actionCANCER RESEARCH, 2016, 76Edgar, Kyle A.论文数: 0 引用数: 0 h-index: 0Song, Kyung论文数: 0 引用数: 0 h-index: 0Schmidt, Stephen论文数: 0 引用数: 0 h-index: 0Kirkpatrick, Don论文数: 0 引用数: 0 h-index: 0Phu, Lilian论文数: 0 引用数: 0 h-index: 0Nannini, Michelle论文数: 0 引用数: 0 h-index: 0Hong, Rebecca论文数: 0 引用数: 0 h-index: 0Cheng, Eric论文数: 0 引用数: 0 h-index: 0Young, Amy论文数: 0 引用数: 0 h-index: 0Sampath, Deepak论文数: 0 引用数: 0 h-index: 0Friedman, Lori S.论文数: 0 引用数: 0 h-index: 0
- [3] Characterization of the enhanced potency of PI3K inhibitor taselisib (GDC-0032) in PI3K mutant cell lines and modelsCANCER RESEARCH, 2015, 75Edgar, Kyle A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USANannini, Michelle论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHong, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAEigenbrot, Charlie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASchmidt, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAYoung, Amy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASampath, Deepak论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWallin, Jeffrey J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAFriedman, Lori S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [4] Determination of the PI3Kα selective inhibitor alpelisib mechanism of action and efficacy in ER+/ PIK3CA mutant breast cancer preclinical modelsCANCER RESEARCH, 2018, 78 (13)Fritsch, Christine论文数: 0 引用数: 0 h-index: 0机构: Novartis AG, Basel, Switzerland Novartis AG, Basel, SwitzerlandPfister, Estelle论文数: 0 引用数: 0 h-index: 0机构: Novartis AG, Basel, Switzerland Novartis AG, Basel, SwitzerlandEbel, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Novartis AG, Basel, Switzerland Novartis AG, Basel, SwitzerlandGuthy, Daniel论文数: 0 引用数: 0 h-index: 0机构: Novartis AG, Basel, Switzerland Novartis AG, Basel, SwitzerlandSchnell, Christian论文数: 0 引用数: 0 h-index: 0机构: Novartis AG, Basel, Switzerland Novartis AG, Basel, SwitzerlandHofmann, Francesco论文数: 0 引用数: 0 h-index: 0机构: Novartis AG, Basel, Switzerland Novartis AG, Basel, Switzerland
- [5] Dual PI3K/mTOR inhibition in PIK3CA mutant pancreatic cancersCANCER RESEARCH, 2018, 78 (13)Payne, Susan论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USADepke, Mitchell论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USAYueh, Alex论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USASharick, Joseph T.论文数: 0 引用数: 0 h-index: 0机构: Morgridge Inst Res, Madison, WI USA Univ Wisconsin, Madison, WI USAFavreau, Peter F.论文数: 0 引用数: 0 h-index: 0机构: Morgridge Inst Res, Madison, WI USA Univ Wisconsin, Madison, WI USAPasch, Cheri A.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USAClipson, Linda论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USAMatkowskyj, Kristina A.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USASkala, Melissa论文数: 0 引用数: 0 h-index: 0机构: Morgridge Inst Res, Madison, WI USA Univ Wisconsin, Madison, WI USADeming, Dustin A.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Madison, WI USA Univ Wisconsin, Madison, WI USA
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- [7] Aspirin has a better effect on PIK3CA mutant colorectal cancer cells by PI3K/Akt/Raptor pathwayMolecular Medicine, 2020, 26Zhihang Chen论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal SurgeryChun Wang论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal SurgeryHao Dong论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal SurgeryXing Wang论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal SurgeryFeng Gao论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal SurgerySen Zhang论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal SurgeryXiaolong Zhang论文数: 0 引用数: 0 h-index: 0机构: the First Affiliated Hospital,Department of Colorectal and Anal Surgery
- [8] Aspirin has a better effect on PIK3CA mutant colorectal cancer cells by PI3K/Akt/Raptor pathwayMOLECULAR MEDICINE, 2020, 26 (01)Chen, Zhihang论文数: 0 引用数: 0 h-index: 0机构: Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R ChinaWang, Chun论文数: 0 引用数: 0 h-index: 0机构: Wuhan Univ, Dept Gastroenterol, Zhongnan Hosp, Wuhan 430000, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R ChinaDong, Hao论文数: 0 引用数: 0 h-index: 0机构: Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R ChinaWang, Xing论文数: 0 引用数: 0 h-index: 0机构: Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R ChinaGao, Feng论文数: 0 引用数: 0 h-index: 0机构: Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R ChinaZhang, Sen论文数: 0 引用数: 0 h-index: 0机构: Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R ChinaZhang, Xiaolong论文数: 0 引用数: 0 h-index: 0机构: Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China Guangxi Med Univ, Affiliated Hosp 1, Dept Colorectal & Anal Surg, Nanning 530021, Peoples R China
- [9] Phase I evaluation of the PI3 kinase (PI3K) inhibitor taselisib (GDC-0032) in multiple locally advanced or metastatic PIK3CA mutant solid tumor types.JOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (15)Jhaveri, Komal L.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABedard, Philippe L.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USACejalvo, Juan Miguel论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHart, Lowell L.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAJuric, Dejan论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAKelly, Karen论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALockhart, A. Craig论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMelnyk, Anton论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMoore, Kathleen N.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USANemunaitis, John J.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAOliveira, Mafalda论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAPatel, Manish R.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USASachdev, Jasgit论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USASmith, David论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAVanderWalde, Ari论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWare, Joseph A.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAJin, Huan论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWilson, Timothy R.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWei, Michael C.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABaselga, Jose论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA
- [10] Differential response to a dual PI3K/mTOR inhibitor in PIK3CA mutant urothelial cancer patient derived xenograftsCANCER RESEARCH, 2016, 76Elbanna, May F.论文数: 0 引用数: 0 h-index: 0Ciamporcero, Eric论文数: 0 引用数: 0 h-index: 0Adelaiye, Remi论文数: 0 引用数: 0 h-index: 0Orillion, Ashley论文数: 0 引用数: 0 h-index: 0Chintala, Sreenivasulu论文数: 0 引用数: 0 h-index: 0Pili, Roberto论文数: 0 引用数: 0 h-index: 0