4-aryl-2,4-dioxobutanoic acid inhibitors of HIV-1 integrase and viral replication in cells

被引：221

作者：

Wai, JS

Egbertson, MS

Payne, LS

Fisher, TE

Embrey, MW

Tran, LO

Melamed, JY

Langford, HM

Guare, JP

Zhuang, LG

Grey, VE

Vacca, JP

Holloway, MK

Naylor-Olsen, AM

Hazuda, DJ

Felock, PJ

Wolfe, AL

Stillmock, KA

Schleif, WA

Gabryelski, LJ

Young, SD

机构：

[1] Merck Res Labs, Dept Med Chem, W Point, PA 19486 USA

[2] Merck Res Labs, Dept Mol Syst, W Point, PA 19486 USA

[3] Merck Res Labs, Dept Antiviral Res, W Point, PA 19486 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 26期

关键词：

D O I：

10.1021/jm000176b

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：4923 / 4926

页数：4

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