Interfacing Chemical Biology and Drug Discovery: Report from the 50th International Conference on Medicinal Chemistry of the SCT (French Medicinal Chemistry Society), July 2-4, 2014, Rouen, France

被引:1
作者
Sapi, Janos [1 ]
Schmidt, Frederic [2 ]
Van Hijfte, Luc [3 ]
George, Pascal [4 ]
机构
[1] Univ Reims, UMR CNRS 7312, SCT, F-51069 Reims, France
[2] Inst Curie, Res Ctr, CNRS UMR3666, INSERM U1143,SCT, F-75248 Paris, France
[3] NovAliX, F-67405 Illkirch Graffenstaden, France
[4] SCT, F-78730 Longvilliers, France
关键词
INHIBITOR TAK-632; OPTIMIZATION; DESIGN; POTENT; IDENTIFICATION; PEPTIDES; PRODRUG; GROWTH;
D O I
10.1021/cb5009469
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:2702 / 2707
页数:6
相关论文
共 54 条
  • [51] Oxetanes in Drug Discovery: Structural and Synthetic Insights
    Wuitschik, Georg
    Carreira, Erick M.
    Wagner, Bjoern
    Fischer, Holger
    Parrilla, Isabelle
    Schuler, Franz
    Rogers-Evans, Mark
    Mueller, Klaus
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (08) : 3227 - 3246
  • [52] Natural Product-Like Macrocyclic N-Methyl-Peptide Inhibitors against a Ubiquitin Ligase Uncovered from a Ribosome-Expressed De Novo Library
    Yamagishi, Yusuke
    Shoji, Ikuo
    Miyagawa, Shoji
    Kawakami, Takashi
    Katoh, Takayuki
    Goto, Yuki
    Suga, Hiroaki
    [J]. CHEMISTRY & BIOLOGY, 2011, 18 (12): : 1562 - 1570
  • [53] Diastereomeric Spirooxindoles as Highly Potent and Efficacious MDM2 Inhibitors
    Zhao, Yujun
    Liu, Liu
    Sun, Wei
    Lu, Jianfeng
    McEachern, Donna
    Li, Xiaoqin
    Yu, Shanghai
    Bernard, Denzil
    Ochsenbein, Philippe
    Ferey, Vincent
    Carry, Jean-Christophe
    Deschamps, Jeffrey R.
    Sun, Duxin
    Wang, Shaomeng
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2013, 135 (19) : 7223 - 7234
  • [54] Total Synthesis of (-)-Zampanolide and Structure-Activity Relationship Studies on (-)-Dactylolide Derivatives
    Zurwerra, Didier
    Glaus, Florian
    Betschart, Leo
    Schuster, Julia
    Gertsch, Juerg
    Ganci, Walter
    Altmann, Karl-Heinz
    [J]. CHEMISTRY-A EUROPEAN JOURNAL, 2012, 18 (52) : 16868 - 16883