共 52 条
Inhibitory effects of transcription factor Ikaros on the expression of liver cancer stem cell marker CD133 in hepatocellular carcinoma
被引:37
作者:

Zhang, Lin
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机构:
Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Li, Hong
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h-index: 0
机构:
Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Ge, Chao
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h-index: 0
机构:
Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Li, Meng
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h-index: 0
机构:
Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Zhao, Fang-yu
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Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Hou, He-lei
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Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Zhu, Miao-xin
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Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Tian, Hua
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Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Zhang, Li-xing
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Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Chen, Tao-yang
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机构:
Qi Dong Liver Canc Inst, Qi Dong, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Jiang, Guo-ping
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机构:
Zhejiang Univ, Sch Med, Affiliated Hosp 1, Dept Gen Surg, Hangzhou 310003, Zhejiang, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Xie, Hai-yang
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机构:
Zhejiang Univ, Sch Med, Affiliated Hosp 1, Dept Gen Surg, Hangzhou 310003, Zhejiang, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Cui, Ying
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h-index: 0
机构:
Canc Inst Guangxi, Nanning, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Yao, Ming
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h-index: 0
机构:
Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China

Li, Jin-jun
论文数: 0 引用数: 0
h-index: 0
机构:
Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China
机构:
[1] Shanghai Jiao Tong Univ, Sch Med, State Key Lab Oncogenes & Related Genes, Shanghai Canc Inst,Renji Hosp, Shanghai 200030, Peoples R China
[2] Qi Dong Liver Canc Inst, Qi Dong, Peoples R China
[3] Zhejiang Univ, Sch Med, Affiliated Hosp 1, Dept Gen Surg, Hangzhou 310003, Zhejiang, Peoples R China
[4] Canc Inst Guangxi, Nanning, Peoples R China
来源:
基金:
中国国家自然科学基金;
关键词:
Ikaros;
CD133;
hepatocellular carcinoma;
cancer stem cells;
TUMOR-INITIATING CELLS;
GROWTH-FACTOR-BETA;
STEM/PROGENITOR CELLS;
EPIGENETIC REGULATION;
COREPRESSOR CTBP;
PROSTATE-CANCER;
DNA-BINDING;
IN-VITRO;
GENE;
ACTIVATION;
D O I:
10.18632/oncotarget.2524
中图分类号:
R73 [肿瘤学];
学科分类号:
100214 ;
摘要:
CD133 is a cellular surface glycoprotein that has been reported as a marker for the enrichment of cancer stem cells (CSCs). However, the regulatory mechanism of CD133 remains unknown. CSCs have been proposed to contribute to radioresistance and multi-drug resistance. The elucidation of key regulators of CD133 and CSCs is critical for the development of CSC-targeted therapy. In this study, we showed that Ikaros inhibited the expression of CD133 via direct binding to the CD133 P1 promoter and repressed the tumorigenic and self-renewal capacity of CD133(+) cancer stem-like cells in hepatocellular carcinoma (HCC). We found that Ikaros interacted with CtBP as a transcription repressor complex, which inhibited CD133 expression in HCC. We also demonstrated that Ikaros expression was up-regulated by ETS1 which activity was regulated by MAPKs pathway. Furthermore, decreased expression of Ikaros was significantly associated with poor survival in HCC patients. Overall, our study identifies that Ikaros plays a role as a transcription repressor in HCC and is a new reactivated therapeutic target for the treatment of HCC. Meanwhile, our findings provide evidence that Ikaros could be an attractive inhibitor of the target gene CD133, which reactivates anticancer mechanisms in targeted CSC therapy.
引用
收藏
页码:10621 / 10635
页数:15
相关论文
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机构:
Zhejiang Univ, Sch Med, Affiliated Hosp 1, Dept Gen Surg, Hangzhou 310003, Zhejiang, Peoples R China Jiao Tong Univ, Shanghai Canc Inst, State Key Lab Oncogenes & Related Genes, Shanghai 200032, Peoples R China

Gu, Jianren
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h-index: 0
机构:
Jiao Tong Univ, Shanghai Canc Inst, State Key Lab Oncogenes & Related Genes, Shanghai 200032, Peoples R China Jiao Tong Univ, Shanghai Canc Inst, State Key Lab Oncogenes & Related Genes, Shanghai 200032, Peoples R China
[20]
Expression and possible role of ets-1 in hepatocellular carcinoma
[J].
Ito, Y
;
Miyoshi, E
;
Takeda, T
;
Sakon, M
;
Noda, K
;
Tsujimoto, M
;
Monden, M
;
Taniguchi, N
;
Matsuura, N
.
AMERICAN JOURNAL OF CLINICAL PATHOLOGY,
2000, 114 (05)
:719-725

Ito, Y
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Miyoshi, E
论文数: 0 引用数: 0
h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Takeda, T
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Sakon, M
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Noda, K
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Tsujimoto, M
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Monden, M
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Taniguchi, N
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan

Matsuura, N
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h-index: 0
机构: Osaka Univ, Sch Allied Hlth Sci, Fac Med, Dept Pathol, Osaka 5650871, Japan