Design, Synthesis, and Biological Screening of Novel Anthranilic Diamides

被引：8

作者：

Hua, Xuewen ^{[1
,2
]}

Mao, Wutao ^{[2
,3
]}

Fan, Zhijin ^{[1
,2
]}

Ji, Xiaotian ^{[1
,2
]}

Li, Fengyun ^{[1
,2
]}

Zong, Guangning ^{[1
,2
]}

Song, Haibin ^{[1
]}

Tatiana, Kalinina ^{[4
]}

Morzherin, Yury Yu. ^{[4
]}

Belskaya, Nataliya P. ^{[4
]}

Bakulev, Vasiliy A. ^{[4
]}

机构：

[1] Nankai Univ, State Key Lab Elementoorgan Chem, 94 Weijin Rd, Tianjin 300071, Peoples R China

[2] Collaborat Innovat Ctr Chem Sci & Engn Tianjin, Tianjin 300071, Peoples R China

[3] Nanyang Normal Univ, Coll Chem & Pharm Engn, Nanyang 473061, Henan, Peoples R China

[4] Ural Fed Univ, Ekaterinburg 620002, Russia

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2016年 / 53卷 / 03期

基金：

对外科技合作项目（国际科技项目）;

关键词：

INSECTICIDES; DERIVATIVES; SULFOXAFLOR; MODE;

D O I：

10.1002/jhet.2351

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Three series of new anthranilic diamide derivatives containing sulfide, N-cyanomethylsulfilimine, and N-cyanomethylsulfoximine groups were designed and synthesized by combining the active substructures of anthranilic diamides and sulfoxaflor. The structures of all newly synthesized compounds were confirmed by IR and H-1/C-13-NMR, and some of them were confirmed by elemental analysis or HRMS too. The synthesized compounds were screened for their insecticidal and fungicidal activities. Bioasssay results indicated that some of the synthesized compounds possessed certain degrees of insecticidal activity against Mythimna separata. However, some compounds exhibited good fungicidal activity against Sclerotinia sclerotiorum.

引用

页码：865 / 875

页数：11

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