Synthesis of ecteinascidin ET-743 and phthalascidin Pt-650 from cyanosafracin B

被引：241

作者：

Cuevas, C ^{[1
]}

Pérez, M ^{[1
]}

Martín, MJ ^{[1
]}

Chicharro, JL ^{[1
]}

Fernández-Rivas, C ^{[1
]}

Flores, M ^{[1
]}

Francesch, A ^{[1
]}

Gallego, P ^{[1
]}

Zarzuelo, M ^{[1
]}

de la Calle, F ^{[1
]}

García, J ^{[1
]}

Polanco, C ^{[1
]}

Rodríguez, I ^{[1
]}

Manzanares, I ^{[1
]}

机构：

[1] Pharma Mar, Madrid 28760, Spain

来源：

ORGANIC LETTERS | 2000年 / 2卷 / 16期

关键词：

D O I：

10.1021/ol0062502

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[GRAPHICS] An efficient new process is described for the synthesis of ecteinascidin ET-743 (1) and phthalascidin (2), starting from readily available cyanosafracin B (3).

引用

页码：2545 / 2548

页数：4

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