A convenient synthesis of 3-amino-4-imino(thioxo)-imidazolidin-2-ones

被引：14
作者：
Kurz, T [1 ]
Widyan, K [1 ]
机构：
[1] Univ Hamburg, Inst Pharm, D-20146 Hamburg, Germany
来源：
TETRAHEDRON LETTERS | 2004年 / 45卷 / 38期
关键词：
diethylphosphonopropyl alpha-aminonitriles; 1,1 '-carbonyldiimidazole; 1,1 '-carbonyl-di-(1,2,4-triazole); hydrazines; 3-amino-4imino(thioxo)-imidazolidin-2-ones;
D O I：
10.1016/j.tetlet.2004.07.134
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Subsequent treatment of diethylphosphonopropyl alpha-aminonitriles with 1,1'-carbonyldiimidazole or 1,1'-carbonyl-di(1,2,4-triazole) and hydrazines afforded substituted 3-amino-4-imino-imidazolidin-2-ones. Their acidic hydrolysis and their reactions with hydrogen sulfide are described. (C) 2004 Elsevier Ltd. All rights reserved.
引用
收藏
页码：7049 / 7051
页数：3
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