BRD4 Degradation By Protacs Represents a More Effective Therapeutic Strategy Than BRD4 Inhibitors in DLBCL

被引:0
作者
Lu, Jing [1 ]
Qian, Yimin [1 ]
Raina, Kanak [1 ]
Altieri, Martha [1 ]
Dong, Hanqing [1 ]
Wang, Jing [1 ]
Chen, Xin [1 ]
Crew, Andrew [1 ]
Coleman, Kevin [1 ]
Crews, Craig [2 ]
Winkler, James [1 ]
机构
[1] Arvinas LLC, New Haven, CT USA
[2] Yale Univ, Dept Mol Cellular & Dev Biol, Dept Chem, Dept Pharmacol, New Haven, CT USA
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R5 [内科学];
学科分类号
1002 ; 100201 ;
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页数:3
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