Heteroannulated Quinazoline and Quinazolinone Derivatives from (Z)-2-[1-Benzamido-2-(3,4,5-trimethoxyphenyl)]vinyl-3,1-benzoxazin-4(3H)-one

被引：7

作者：

Mahmoud, Mahmoud R. ^{[1
]}

Derbala, Hamed A. Y. ^{[1
]}

机构：

[1] Ain Shams Univ, Fac Sci, Dept Chem, Cairo, Egypt

来源：

SYNTHETIC COMMUNICATIONS | 2010年 / 40卷 / 10期

关键词：

Benzoxazin-4(3H)-one; imidazo-[1; 5-b]-quinazolin-4(3H)-one derivatives; 1; 2; 5]-oxadiazino-[3; 2-b]-quinazolin-4(3H)-one derivatives; 4]-triazino-[6; 1-b]-quinazolin-4(3H)-one derivatives; 4]-triazolo-[1; 5-c]-quinazolin-4(3H)-one derivatives; FACILE SYNTHESIS; 4(3H)-QUINAZOLINONE DERIVATIVES; BIOLOGICAL EVALUATION; INHIBITORS; 3-AMINO-2(1H)-THIOXO-4(3H)-QUINAZOLINONE; ANALOGS;

D O I：

10.1080/00397910903098722

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The title compound 1 was prepared and allowed to react with a series of nitrogen nucleophiles to afford the quinazoline and quinazolinone derivatives 2-12 and tetrazole derivative 13. The IR, 1H NMR, 13C NMR, and mass spectra of all the synthesized compounds were discussed.

引用

收藏

页码：1516 / 1529

页数：14

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